GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ALPG |
N-[3-(methylthio)phenyl]-3-phenylacrylamide |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
N-(3-chloro-2-methylphenyl)-N'-cyclohexylurea |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-[2-(Dimethylamino)-1-propenyl]-3-nitro-1-benzofuran-5-ol |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-(5-phenyl-1H-1,2,4-triazol-3-yl)-3a,4,7,7a-tetrahydroisoindole-1,3-quinone |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
3-(Benzothiazol-2-ylsulfanylmethyl)-6-chloro-3H-benzooxazol-2-one |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
2-(5-benzyl-1H-1,2,4-triazol-3-yl)-3a,4,7,7a-tetrahydroisoindole-1,3-quinone |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
6-Amino-4-(4-hydroxy-3,5-dimethoxy-phenyl)-3-(methoxymethyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
(6E)-2-methoxy-6-[([1,2,4]triazolo[3,4-a]phthalazin-6-ylhydrazo)methylidene]-1-cyclohexa-2,4-dienone |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
6-Amino-4-(4-hydroxy-3-methoxy-phenyl)-3-propyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
Dimorpholinophosphoryl(piperidino)methanone oxime |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
(5E)-4-keto-2-methyl-5-vanillylidene-2-pyrroline-3-carboxylic acid methyl ester |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
(2Z)-2-[(3-methoxy-4-oxidanyl-phenyl)methylidene]-6,7,8,9-tetrahydro-5H-imidazo[1,2-a]azepin-3-one |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
3-[1-[(4-Nitrophenyl)hydrazinylidene]ethyl]aniline |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
[(2-Chlorobenzylidene)amino]-(2-nitrophenyl)amine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
5-Chloro-2-(1-naphthylmethoxy)benzaldoxime |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
N-[(3-chloro-2-piperidin-1-ylphenyl)carbamothioyl]butanamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1-(4-methylphenyl)-N-(thiophen-2-ylmethyl)benzimidazol-5-amine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
7-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo[4,3-c]pyrimidine |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
3-(1H-benzimidazol-2-yl)-1-[4-(2,4-dimethylphenyl)-1-piperazinyl]-1-propanone |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-(4-fluorobenzyl)-2-(2-keto-6-pyrrolidinosulfonyl-1,3-benzoxazol-3-yl)acetamide |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |