GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ALPPL2 |
6-Phosphonohexanoic acid |
7000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
Phenylsulfanylmethyl-phosphonothioic acid |
460000 |
NA |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
6-Thiophosphono-hexanoic acid methyl ester |
330000 |
NA |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
Benzyl-phosphonothioic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
6-Thiophosphono-hexanoic acid |
1500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
11-Oxo-11 h-pyrido[2,1-b]quinazoline-7-carboxylic acid |
NA |
170000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
12-oxo-12H-benzo[g]pyrido[2,1-b]quinazoline-4-carboxylic acid |
NA |
710000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
2-Hydroxy-11-oxopyrido[2,1-b]quinazoline-8-carboxylic acid |
NA |
280000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
2,3-Dimethoxy-11-oxo-11H-pyrido[2,1-b]quinazoline-8-carboxylic acid |
NA |
410000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
2,3-Dihydroxy-11-oxopyrido[2,1-b]quinazoline-8-carboxylic acid |
NA |
220000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
3-methoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one |
NA |
620000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
2-(2H-tetrazol-5-yl)-12H-benzo[g]pyrido[2,1-b]quinazolin-12-one |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
2-methoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one |
NA |
280000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
2-methyl-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one |
NA |
210000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
2,3-dimethoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one |
NA |
340000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
6-(2H-tetrazol-5-yl)-13,15-dioxa-2,8-diazatetracyclo[8.7.0.03,8.012,16]heptadeca-1(17),2,4,6,10,12(16)-hexaen-9-one |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
Zaprinast |
NA |
6250000 |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
Methylphosphonic acid |
11000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
Methylphosphonothiolate |
19000000 |
NA |
NA |
NA |
NA |
NA |
TTD |