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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ALPPL2 6-Phosphonohexanoic acid 7000000 NA NA NA NA NA TTD
ALPPL2 Phenylsulfanylmethyl-phosphonothioic acid 460000 NA NA NA NA NA TTD
ALPPL2 6-Thiophosphono-hexanoic acid methyl ester 330000 NA NA NA NA NA TTD
ALPPL2 Benzyl-phosphonothioic acid 200000 NA NA NA NA NA TTD
ALPPL2 6-Thiophosphono-hexanoic acid 1500000 NA NA NA NA NA TTD
ALPPL2 11-Oxo-11 h-pyrido[2,1-b]quinazoline-7-carboxylic acid NA 170000 NA NA NA NA TTD
ALPPL2 12-oxo-12H-benzo[g]pyrido[2,1-b]quinazoline-4-carboxylic acid NA 710000 NA NA NA NA TTD
ALPPL2 2-Hydroxy-11-oxopyrido[2,1-b]quinazoline-8-carboxylic acid NA 280000 NA NA NA NA TTD
ALPPL2 2,3-Dimethoxy-11-oxo-11H-pyrido[2,1-b]quinazoline-8-carboxylic acid NA 410000 NA NA NA NA TTD
ALPPL2 2,3-Dihydroxy-11-oxopyrido[2,1-b]quinazoline-8-carboxylic acid NA 220000 NA NA NA NA TTD
ALPPL2 3-methoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one NA 620000 NA NA NA NA TTD
ALPPL2 2-(2H-tetrazol-5-yl)-12H-benzo[g]pyrido[2,1-b]quinazolin-12-one NA 230000 NA NA NA NA TTD
ALPPL2 2-methoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one NA 140000 NA NA NA NA TTD
ALPPL2 8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one NA 280000 NA NA NA NA TTD
ALPPL2 2-methyl-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one NA 210000 NA NA NA NA TTD
ALPPL2 2,3-dimethoxy-8-(2H-tetrazol-5-yl)pyrido[2,1-b]quinazolin-11-one NA 340000 NA NA NA NA TTD
ALPPL2 6-(2H-tetrazol-5-yl)-13,15-dioxa-2,8-diazatetracyclo[8.7.0.03,8.012,16]heptadeca-1(17),2,4,6,10,12(16)-hexaen-9-one NA 230000 NA NA NA NA TTD
ALPPL2 Zaprinast NA 6250000 NA NA NA NA TTD
ALPPL2 Methylphosphonic acid 11000000 NA NA NA NA NA TTD
ALPPL2 Methylphosphonothiolate 19000000 NA NA NA NA NA TTD