| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ALPPL2 |
11-Oxo-11H-pyrido(2,1-b)quinazoline-8-carboxylic acid |
NA |
350000 |
NA |
NA |
NA |
NA |
TTD |
| ALPPL2 |
Butyl-phosphonothioic acid |
600000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ALPPL2 |
Propylphosphonic acid |
1550000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ALPPL2 |
4-Oxopyrido[1,2-a]pyrimidine-7-carboxylic acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| ALPPL2 |
Cromolyn Sodium |
NA |
9680000 |
NA |
NA |
NA |
NA |
TTD |
| ALPPL2 |
2-Methyl-11-oxo-11H-pyrido(2,1-b)quinazoline-8-carboxylic acid |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| ALPPL2 |
12H-Benzo(g)pyrido(2,1-b)quinazoline-2-carboxylic acid, 12-oxo- |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| ALPPL2 |
2,3,4,11-tetrahydro-1H-pyrido[2,1-b]quinazoline-8-carboxylic acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| ALPPL2 |
11-Oxo-11H-pyrido[2,1-b]quinazoline-6-carboxylic acid |
NA |
800000 |
NA |
NA |
NA |
NA |
TTD |
| ALPPL2 |
Bufrolin |
NA |
970000 |
NA |
NA |
NA |
NA |
TTD |
| ALPPL2 |
Benzylphosphonic Acid |
580000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
4-N-[3,5-bis(trifluoromethyl)phenyl]-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
4-N-(3,5-dichlorophenyl)pyridine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
4-N-(3-chloro-5-fluorophenyl)-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
4-N-(3,5-dichloro-4-fluorophenyl)-6-methylpyrimidine-2,4-diamine |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
4-N-(3,5-dichlorophenyl)-6-(trifluoromethyl)pyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl-[(3R,5S)-5-carboxypyrrolidin-3-yl]-methylsulfanium;hydrogen sulfate;sulfuric acid |
1070000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
(3-amino-3-cyanopropyl)-[[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl]-methylsulfanium;bromide;hydrobromide |
246600 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| AMD1 |
[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl-methyl-pyrrolidin-3-ylsulfanium;hydrogen sulfate;sulfuric acid |
669000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| AMD1 |
[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl-[(5S)-5-carboxypyrrolidin-3-yl]-methylsulfanium;hydrogen sulfate;sulfuric acid |
1070000|1207000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |