GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
AMD1 |
N-(3,5-dichlorophenyl)-6-methylpyrimidin-4-amine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-(3-bromo-5-ethylphenyl)-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-(3,5-Dichlorophenyl)sulfanyl-6-methylpyrimidin-2-amine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-(3-chloro-5-pyrimidin-5-ylphenyl)-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-(3,5-diphenylphenyl)-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-[3-chloro-5-(3-chloro-4-fluorophenyl)phenyl]-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-(3-chloro-5-phenanthren-9-ylphenyl)-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
5-[(2-amino-6-methylpyrimidin-4-yl)amino]-1-N,3-N-bis(3,5-dichlorophenyl)benzene-1,3-dicarboxamide |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-[3-ethyl-5-(4-fluorophenyl)phenyl]-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-[3-chloro-5-(2-chlorophenyl)phenyl]-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-[3-chloro-5-(3,4-dichlorophenyl)phenyl]-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-[3-(2,1,3-benzoxadiazol-5-yl)-5-chlorophenyl]-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-(3,5-dichlorophenyl)-2-N,2-N,6-trimethylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-[(2-Amino-6-methylpyrimidin-4-yl)amino]-2,6-dichlorophenol |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-[3-bromo-5-(2-methylpropoxy)phenyl]-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-[3-[3,5-bis(trifluoromethyl)phenyl]-5-chlorophenyl]-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-[3-[(2-Amino-6-methylpyrimidin-4-yl)amino]-5-chlorophenyl]phenol |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-[3-chloro-5-[4-chloro-3-(trifluoromethyl)phenyl]phenyl]-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
5-[(2-Amino-6-methylpyrimidin-4-yl)amino]benzene-1,3-dicarboxylic acid |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-[3-chloro-5-(3-chlorophenyl)phenyl]-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |