| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| AMD1 |
(2R,3R,4S,5R)-2-(6-amino-8-ethylpurin-9-yl)-5-[[3-aminopropyl(methyl)amino]methyl]oxolane-3,4-diol;sulfuric acid |
NA |
420000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
6-Methyl-N4-(o-tolyl)pyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
Methyl 3-((2-amino-6-methylpyrimidin-4-yl)amino)-5-(methoxycarbonyl)benzoate |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
N~4~-(3-fluorophenyl)-6-methyl-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
6-methyl-N~4~-[2-(methylthio)phenyl]-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
N~4~-(4-bromo-2-fluorophenyl)-6-methyl-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
N~4~-(3,4-difluorophenyl)-6-methyl-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
2-Amino-4-(3-bromophenyl)amino-6-methylpyrimidine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
N~4~-(5-chloro-2-methylphenyl)-6-methyl-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
N~4~-(4-chloro-2-methylphenyl)-6-methyl-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
N~4~-[2-chloro-5-(trifluoromethyl)phenyl]-6-methyl-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
N~4~-(4-ethylphenyl)-6-methyl-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
N~4~-(3-chloro-2-methylphenyl)-6-methyl-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
6-methyl-N~4~-[4-(trifluoromethyl)phenyl]-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
N~4~-(2,3-dichlorophenyl)-6-methyl-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
N~4~-(2,4-dichlorophenyl)-6-methyl-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
N~4~-(4-isopropylphenyl)-6-methyl-2,4-pyrimidinediamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
2-Amino-4-phenylamino-6-methylpyrimidine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
2-N-(3,5-dichlorophenyl)pyridine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| AMD1 |
6-N-(3,5-dichlorophenyl)pyridine-2,6-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |