| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| AMY1A |
|
NA |
330000 |
NA |
NA |
NA |
NA |
BindingDB |
| AMY1A |
4-{2-[(4-Hydroxyphenyl)amino]-1,3-thiazol-4-yl}phenol |
NA |
492000 |
NA |
NA |
NA |
NA |
BindingDB |
| AMY1A |
4-N-[4-(2,4-dichlorophenyl)-1,3-thiazol-2-yl]benzene-1,4-diamine |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB |
| AMY1B |
Epigallocatechin Gallate |
NA |
1400000 |
NA |
NA |
NA |
NA |
PubChem |
| AMY1C |
Epigallocatechin Gallate |
NA |
1400000 |
NA |
NA |
NA |
NA |
PubChem |
| AMY2A |
D-Gluconhydroximo-1,5-Lactam |
18000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AMY2A |
Maltosyl-Alpha (1,4)-D-Gluconhydroximo-1,5-Lactam |
1800000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ANG |
rAdo-P-P-dUrd |
360000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ANG |
Adenylate-3'-phosphate-((2'-deoxy-uridine-5'-phosphate)-3'-phosphate) |
360000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ANG |
2-amino-3-hydroxy-N-[(2S,3R,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]propanamide |
427000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ANG |
2-amino-N-[(2S,3R,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]-3-(4-hydroxyphenyl)propanamide |
1251000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ANG |
2-[[(2S,3R,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]amino]-2-oxoacetic acid |
775000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ANG |
3-[[(2S,3R,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]amino]-3-oxopropanoic acid |
1114000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ANPEP |
2-[2,6-bis(propan-2-yl)phenyl]-3-sulfanylidene-2,3-dihydro-1H-isoindol-1-one |
NA |
309200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(S)-2-((1R,2S)-2-Amino-1-carbamoyl-3-phenyl-propylamino)-4-methyl-pentanoic acid methyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
4-Amino-2-(2,6-dimethyl-phenyl)-isoindole-1,3-dione |
NA |
108000|108900 |
NA |
NA |
NA |
NA |
BindingDB |
| ANPEP |
2-(2,6-Dimethyl-phenyl)-4-hydroxy-isoindole-1,3-dione |
NA |
264000|264500|265000 |
NA |
NA |
NA |
NA |
BindingDB |
| ANPEP |
2-(2,4-dimethylphenyl)-4H-isoquinoline-1,3-dione |
NA |
188000 |
NA |
NA |
NA |
NA |
BindingDB |
| ANPEP |
2-(2-propan-2-ylphenyl)-4H-isoquinoline-1,3-dione |
NA |
193000 |
NA |
NA |
NA |
NA |
BindingDB |
| ANPEP |
(2S,4S)-Methyl 1-acetyl-4-(benzamido)pyrrolidine-2-carboxylate |
NA |
122500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |