| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ANPEP |
(2S,4S)-Methyl 1-((E)-3-(3,4-dimethoxyphenyl)acryloyl)-4-(nicotinamido)pyrrolidine-2-carboxylate |
NA |
137300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
2-Phenylisoquinoline-1,3(2h,4h)-dione |
NA |
396000 |
NA |
NA |
NA |
NA |
BindingDB |
| ANPEP |
3-Amino-4-phenylbutanoic acid |
NA |
800000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
1-(Toluene-4-sulfonyl)-4-(toluene-4-sulfonyloxy)-pyrrolidine-2-carboxylic acid methyl ester |
NA |
101400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
Phe-Ser-Arg |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(S)-2-((S)-2-tert-Butoxycarbonylamino-1-cyano-3-phenyl-propylamino)-3-methyl-butyric acid methyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
1-[(S)-2-((1R,2S)-2-Amino-1-carbamoyl-3-phenyl-propylamino)-4-methyl-pentanoyl]-pyrrolidine-2-carboxylic acid methyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
1-[(S)-2-((1S,2S)-2-tert-Butoxycarbonylamino-1-cyano-3-phenyl-propylamino)-4-methyl-pentanoyl]-pyrrolidine-2-carboxylic acid methyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(S)-2-((1R,2S)-2-tert-Butoxycarbonylamino-1-cyano-3-phenyl-propylamino)-3-phenyl-propionic acid methyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(S)-2-((1S,2S)-2-tert-Butoxycarbonylamino-1-cyano-3-phenyl-propylamino)-3-phenyl-propionic acid methyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(S)-6-Amino-2-((S)-2-tert-butoxycarbonylamino-1-cyano-3-phenyl-propylamino)-hexanoic acid methyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(S)-2-((1S,2S)-2-Amino-1-cyano-3-phenyl-propylamino)-3-phenyl-propionic acid methyl ester |
NA |
146000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
1-[(S)-2-((1S,2S)-2-Amino-1-carbamoyl-3-phenyl-propylamino)-4-methyl-pentanoyl]-pyrrolidine-2-carboxylic acid methyl ester |
NA |
783000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
1-[(S)-2-((1R,2S)-2-tert-Butoxycarbonylamino-1-cyano-3-phenyl-propylamino)-4-methyl-pentanoyl]-pyrrolidine-2-carboxylic acid methyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(S)-1-Ammonium-3-methyl-butane-1-phosphonic acid anion |
167000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ANPEP |
2-[(Formyl-Hydroxy-Amino)-Methyl]-Heptanoic Acid [1-(2-Hydroxymethyl-Pyrrolidine-1-Carbonyl)-2-Methyl-Propyl]-Amide |
300000|390000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ANPEP |
4-Hydroxy-2-(2-methylsulfanyl-phenyl)-isoindole-1,3-dione |
NA |
133000|133900 |
NA |
NA |
NA |
NA |
BindingDB |
| ANPEP |
1-Aminoethyl-(1-amino-3-methylbutyl)phosphinic acid |
NA |
155000 |
NA |
NA |
NA |
NA |
BindingDB |
| ANPEP |
(1-Amino-2-methylpropyl)-(phenylcarbamoyl)phosphinic acid |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| ANPEP |
4-(3-Phenyl-acryloyloxy)-1-(toluene-4-sulfonyl)-pyrrolidine-2-carboxylic acid methyl ester |
NA |
168600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |