GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ANPEP |
1-[(S)-2-((S)-2-Amino-3-phenyl-propionylamino)-4-methyl-pentanoyl]-pyrrolidine-2-carboxylic acid methyl ester |
NA |
793000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ANPEP |
(5-fluoro-2,4-dioxopyrimidin-1-yl)methyl (2S)-2-[[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanoyl]amino]-4-methylpentanoate;hydrochloride |
NA |
164170 |
NA |
NA |
NA |
NA |
BindingDB |
ANPEP |
2-(2,6-Diethylphenyl)isoindole-1,3-dione |
NA |
304000 |
NA |
NA |
NA |
NA |
BindingDB |
ANPEP |
L-Leucine, L-phenylalanyl- |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ANPEP |
2-(2-{Bis-[4-(ethoxycarbonylmethyl-carbamoyl)-phenoxy]-phosphoryl}-pyrrolidine-1-carbonyl)-pyrrolidinium; chloride |
NA |
104000 |
NA |
NA |
NA |
NA |
BindingDB |
ANPEP |
7-Amino-5,7,8,9-tetrahydrobenzocyclohepten-6-one,6-oxime hydrochloride |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
ANTXR2 |
Chinese gallotannin |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
ANTXR2 |
3,4-Dihydroxyphenylpropionic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
ANTXR2 |
Gallic Acid |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
ANTXR2 |
Propyl Gallate |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
ANTXR2 |
Quercetin |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
ANTXR2 |
(1E,4Z,6E)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
ANTXR2 |
Dopamine |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
ANTXR2 |
Caffeic Acid |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
ANTXR2 |
Epicatechin |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
ANTXR2 |
Epigallocatechin |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
ANTXR2 |
Vanillic Acid |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
AOC1 |
4-{[4-(Aminomethyl)-5-(4-hydroxybutoxy)pyridin-3-yl]oxy}butan-1-ol dihydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
AOC1 |
[3-(Benzyloxy)-5-ethoxypyridin-4-yl]methylamine dihydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
AOC1 |
4-Pyridinemethanamine, 3,5-diethoxy- |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |