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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ANPEP 1-[(S)-2-((S)-2-Amino-3-phenyl-propionylamino)-4-methyl-pentanoyl]-pyrrolidine-2-carboxylic acid methyl ester NA 793000 NA NA NA NA BindingDB|TTD
ANPEP (5-fluoro-2,4-dioxopyrimidin-1-yl)methyl (2S)-2-[[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanoyl]amino]-4-methylpentanoate;hydrochloride NA 164170 NA NA NA NA BindingDB
ANPEP 2-(2,6-Diethylphenyl)isoindole-1,3-dione NA 304000 NA NA NA NA BindingDB
ANPEP L-Leucine, L-phenylalanyl- NA 1000000 NA NA NA NA BindingDB|TTD
ANPEP 2-(2-{Bis-[4-(ethoxycarbonylmethyl-carbamoyl)-phenoxy]-phosphoryl}-pyrrolidine-1-carbonyl)-pyrrolidinium; chloride NA 104000 NA NA NA NA BindingDB
ANPEP 7-Amino-5,7,8,9-tetrahydrobenzocyclohepten-6-one,6-oxime hydrochloride NA 110000 NA NA NA NA BindingDB
ANTXR2 Chinese gallotannin NA 300000 NA NA NA NA PubChem
ANTXR2 3,4-Dihydroxyphenylpropionic acid NA 300000 NA NA NA NA PubChem
ANTXR2 Gallic Acid NA 300000 NA NA NA NA PubChem
ANTXR2 Propyl Gallate NA 300000 NA NA NA NA PubChem
ANTXR2 Quercetin NA 300000 NA NA NA NA PubChem
ANTXR2 (1E,4Z,6E)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one NA 300000 NA NA NA NA PubChem
ANTXR2 Dopamine NA 300000 NA NA NA NA PubChem
ANTXR2 Caffeic Acid NA 300000 NA NA NA NA PubChem
ANTXR2 Epicatechin NA 300000 NA NA NA NA PubChem
ANTXR2 Epigallocatechin NA 300000 NA NA NA NA PubChem
ANTXR2 Vanillic Acid NA 300000 NA NA NA NA PubChem
AOC1 4-{[4-(Aminomethyl)-5-(4-hydroxybutoxy)pyridin-3-yl]oxy}butan-1-ol dihydrochloride NA 1000000 NA NA NA NA TTD
AOC1 [3-(Benzyloxy)-5-ethoxypyridin-4-yl]methylamine dihydrochloride NA 1000000 NA NA NA NA TTD
AOC1 4-Pyridinemethanamine, 3,5-diethoxy- NA 1000000 NA NA NA NA TTD