| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ANPEP |
1-Benzenesulfonyl-4-(3-phenyl-acryloyloxy)-pyrrolidine-2-carboxylic acid methyl ester |
NA |
134700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
1-Methanesulfonyl-4-(3-phenyl-acryloyloxy)-pyrrolidine-2-carboxylic acid methyl ester |
NA |
114300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(S)-7-(Toluene-4-sulfonyl)-1,4-dioxa-7-aza-spiro[4.4]nonane-8-carboxylic acid methyl ester |
NA |
155800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(S)-2-(Toluene-4-sulfonyl)-6,10-dioxa-2-aza-spiro[4.5]decane-3-carboxylic acid methyl ester |
NA |
173700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
methyl (3S)-2-(4-methylphenyl)sulfonyl-6,11-dioxa-2-azaspiro[4.6]undecane-3-carboxylate |
NA |
124300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
methyl (8S)-7-(benzenesulfonyl)-1,4-dioxa-7-azaspiro[4.4]nonane-8-carboxylate |
NA |
150600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
methyl (3S)-2-(benzenesulfonyl)-6,10-dioxa-2-azaspiro[4.5]decane-3-carboxylate |
NA |
168100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
methyl (3S)-2-(benzenesulfonyl)-6,11-dioxa-2-azaspiro[4.6]undecane-3-carboxylate |
NA |
134800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(3S)-2-(benzenesulfonyl)-N-hydroxy-6,11-dioxa-2-azaspiro[4.6]undecane-3-carboxamide |
NA |
106700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
N-((3S,5S)-1-((E)-3-(3,4-dimethoxyphenyl)acryloyl)-5-(hydroxycarbamoyl)pyrrolidin-3-yl)nicotinamide |
NA |
141900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
Ethyl 2-[[4-[[4-[(2-ethoxy-2-oxoethyl)carbamoyl]phenoxy]-[1-(pyrrolidine-2-carbonyl)pyrrolidin-2-yl]phosphoryl]oxybenzoyl]amino]acetate;hydrochloride |
NA |
104000 |
NA |
NA |
NA |
NA |
TTD |
| ANPEP |
(3S)-3-amino-5-methylhexan-2-one |
430000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
6-Amino-5,6,8,9-tetrahydrobenzocycloheptene-7-one, hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ANPEP |
trans-7-amino-6,7,8,9-tetrahydro-5H-benzocyclohepten-6-ol hydrochloride |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(2R)-2-amino-N-[(2S,3S)-2-amino-3-hydroxy-3-(4-nitrophenyl)propyl]-3-sulfanylpropanamide |
NA |
248350 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(2S)-2-amino-N-[(2R)-1-[[(2S,3S)-2-amino-3-hydroxy-3-(4-nitrophenyl)propyl]amino]-1-oxo-3-phenylpropan-2-yl]-4-methylpentanamide |
NA |
289950 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(2R)-2-amino-N-[(2S)-3-[[(2S,3S)-2-amino-3-hydroxy-3-(4-nitrophenyl)propyl]amino]-2-hydroxy-3-oxopropyl]-3-phenylpropanamide |
NA |
615560 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
H-Phe-Gln-Arg-Phe-Ser-Arg-OH |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
(2S)-N-hydroxy-4-methylsulfanyl-2-(2-phenylethylcarbamoylamino)butanamide |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ANPEP |
Ubenimex |
NA |
471600 |
NA |
NA |
NA |
NA |
PubChem |