| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| AOX1 |
[3,3-Diethoxypropyl(ethoxy)phosphoryl]benzene |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| AOX1 |
[2,2-Diethoxyethyl(ethoxy)phosphoryl]benzene |
400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| AOX1 |
Proadifen |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| AOX1 |
Diethyl (2,2-diethoxyethyl)phosphonate |
1500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| APEX1 |
3-(4-bromothiophen-2-yl)-1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,6H)-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
10-methylpyrimido[4,5-b]quinoline-2,4(3H,10H)-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
1,6-Dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
1,6-Dimethyl-3-(o-tolyl)pyrimido[5,4-e][1,2,4]triazine-5,7(1H,6H)-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
Walrycin B |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
Pyrimido(5,4-e)-1,2,4-triazine-5,7(1H,6H)-dione, 3-(3,4-dimethoxyphenyl)-1,6-dimethyl- |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
3-Methyltoxoflavin |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
1,6-Dimethyl-3-phenylpyrimido[5,4-E][1,2,4]triazine-5,7(1H,6H)-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
3-(4-Chloro-phenyl)-1,6-dimethyl-1H-pyrimido[5,4-e][1,2,4]triazine-5,7-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
1,6-Dimethyl-3-(2-phenylethyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
3-Cyclohexyl-1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
3-Cyclopropyl-1,6-dimethylpyrimido[5,4-e]-1,2,4-triazine-5,7(1H,6H)-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
1-ethyl-3-(4-ethylphenyl)-6-methylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,6H)-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
3-(4-ethylphenyl)-6-methylpyrimido[5,4-e][1,2,4]triazine-5,7(6H,8H)-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
3-benzyl-1,6-dimethyl-1H,5H,6H,7H-pyrimido[5,4-e][1,2,4]triazine-5,7-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| APEX1 |
1,6-Dimethyl-3-(p-tolyl)pyrimido[5,4-e][1,2,4]triazine-5,7(1H,6H)-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |