GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
AMD1 |
4-N-(3,5-difluorophenyl)-6-methylpyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-(3,5-dichlorophenyl)pyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMD1 |
4-N-(3,5-dichlorophenyl)pyrimidine-2,4,6-triamine |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
AMY1A |
4-(2-(4-Hydroxyphenylamino)thiazol-4-yl)benzene-1,3-diol |
NA |
138000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
|
NA |
260000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
(5E)-2-(4-acetylpiperazin-1-yl)-5-(2-hydroxybenzylidene)-1,3-thiazol-4(5H)-one |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
4-{[4-(2,4-Dihydroxyphenyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide |
NA |
165000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
5-{[4-(2,4-Dihydroxyphenyl)-1,3-thiazol-2-yl]amino}-2-hydroxybenzoic acid |
NA |
423000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
|
NA |
4000000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
2-[6-(2-Hydroxy-3-methoxyphenyl)-4,4-dimethyl-3,5-dinitropiperidin-2-yl]-6-methoxyphenol |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
4-{[4-(2,4-Dihydroxyphenyl)-1,3-thiazol-2-yl]amino}-2-hydroxybenzoic acid |
NA |
642000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
1-[2-[[5-(2-Fluorophenyl)furan-2-yl]methylamino]ethylamino]propan-2-ol |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
|
NA |
4000000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
|
NA |
850000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
Epigallocatechin Gallate |
NA |
1400000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
AMY1A |
4-(4-Phenylthiazol-2-ylamino)phenol |
NA |
1274000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
4-{[4-(2,4-Dihydroxyphenyl)-1,3-thiazol-2-yl]amino}benzoic acid |
NA |
680000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
2,6-Bis((2-hydroxy-5-methylphenyl)methyl)-4-methylphenol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
4-[[4-(4-Chlorophenyl)-2-thiazolyl]amino]phenol |
NA |
1043000 |
NA |
NA |
NA |
NA |
BindingDB |
AMY1A |
4-[[4-(4-Methylphenyl)-1,3-thiazol-2-yl]amino]phenol |
NA |
735000 |
NA |
NA |
NA |
NA |
BindingDB |