Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
AMD1 4-N-(3,5-difluorophenyl)-6-methylpyrimidine-2,4-diamine NA 180000 NA NA NA NA TTD
AMD1 4-N-(3,5-dichlorophenyl)pyrimidine-2,4-diamine NA 180000 NA NA NA NA TTD
AMD1 4-N-(3,5-dichlorophenyl)pyrimidine-2,4,6-triamine NA 180000 NA NA NA NA TTD
AMY1A 4-(2-(4-Hydroxyphenylamino)thiazol-4-yl)benzene-1,3-diol NA 138000 NA NA NA NA BindingDB
AMY1A NA 260000 NA NA NA NA BindingDB
AMY1A (5E)-2-(4-acetylpiperazin-1-yl)-5-(2-hydroxybenzylidene)-1,3-thiazol-4(5H)-one NA 700000 NA NA NA NA BindingDB
AMY1A 4-{[4-(2,4-Dihydroxyphenyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide NA 165000 NA NA NA NA BindingDB
AMY1A 5-{[4-(2,4-Dihydroxyphenyl)-1,3-thiazol-2-yl]amino}-2-hydroxybenzoic acid NA 423000 NA NA NA NA BindingDB
AMY1A NA 4000000 NA NA NA NA BindingDB
AMY1A 2-[6-(2-Hydroxy-3-methoxyphenyl)-4,4-dimethyl-3,5-dinitropiperidin-2-yl]-6-methoxyphenol NA 300000 NA NA NA NA BindingDB
AMY1A 4-{[4-(2,4-Dihydroxyphenyl)-1,3-thiazol-2-yl]amino}-2-hydroxybenzoic acid NA 642000 NA NA NA NA BindingDB
AMY1A 1-[2-[[5-(2-Fluorophenyl)furan-2-yl]methylamino]ethylamino]propan-2-ol NA 1000000 NA NA NA NA BindingDB
AMY1A NA 4000000 NA NA NA NA BindingDB
AMY1A NA 850000 NA NA NA NA BindingDB
AMY1A Epigallocatechin Gallate NA 1400000 NA NA NA NA BindingDB|PubChem
AMY1A 4-(4-Phenylthiazol-2-ylamino)phenol NA 1274000 NA NA NA NA BindingDB
AMY1A 4-{[4-(2,4-Dihydroxyphenyl)-1,3-thiazol-2-yl]amino}benzoic acid NA 680000 NA NA NA NA BindingDB
AMY1A 2,6-Bis((2-hydroxy-5-methylphenyl)methyl)-4-methylphenol NA 200000 NA NA NA NA BindingDB
AMY1A 4-[[4-(4-Chlorophenyl)-2-thiazolyl]amino]phenol NA 1043000 NA NA NA NA BindingDB
AMY1A 4-[[4-(4-Methylphenyl)-1,3-thiazol-2-yl]amino]phenol NA 735000 NA NA NA NA BindingDB