GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ALPG |
2-(4-Fluorophenyl)sulfonyl-5-phenyl-3-pyrazolamine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
Octyl(quinazolin-4-yl)amine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
4-[[(3,4-diketo-2-piperidino-cyclobuten-1-yl)amino]methyl]-N-(3,4-dimethoxyphenyl)cyclohexanecarboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
4-[[[3,4-diketo-2-(4-methylpiperidino)cyclobuten-1-yl]amino]methyl]-N-(3,4-dimethoxyphenyl)cyclohexanecarboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-Oxo-2-phenylethyl 2-(propionylamino)benzoate |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
3-(3,4-Dihydroxyphenyl)-2-(phenylsulfonyl)acrylonitrile |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
4-({2-[(4-Fluorobenzyl)oxy]benzyl}amino)benzenesulfonamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
6-[(2-Ethoxyphenoxy)methyl]-3-(4-methylphenyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
N-[3-chloro-4-(difluoromethoxy)phenyl]-3-(difluoromethoxy)benzamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPI |
Levamisole |
NA |
400000|200000 |
NA |
NA |
NA |
NA |
PubChem |
ALPL |
(3Z)-3-[(2-bromophenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
ALPL |
(3Z)-3-[(3-methoxyphenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
ALPL |
(3Z)-3-[(3-bromophenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
ALPL |
(3Z)-3-[(2,4-dichlorophenyl)methylidene]-1,1-dioxo-1lambda6,2-benzothiazin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
ALPL |
(3Z)-3-(3-chlorobenzylidene)-2,3-dihydro-4H-1,2-benzothiazin-4-one 1,1-dioxide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
ALPL |
Phenylalanine |
NA |
100100|200000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
ALPP |
Levamisole |
NA |
400000 |
NA |
NA |
NA |
NA |
PubChem |
ALPP |
Benzylphosphonic Acid |
580000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ALPPL2 |
7-Thiophosphonomethyl-naphthalene-1-carboxylic acid |
1500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
ALPPL2 |
7-Phosphonomethyl-naphthalene-1-carboxylic acid |
390000 |
NA |
NA |
NA |
NA |
NA |
TTD |