| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| APP |
Galangin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| APP |
Ellagic Acid |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| APP |
Anofinic acid |
NA |
NA |
NA |
251500 |
NA |
NA |
BindingDB|TTD |
| APP |
Phenethyl Cinnamate |
NA |
NA |
NA |
1040000 |
NA |
NA |
BindingDB|TTD |
| APP |
Grifolin |
NA |
148800 |
NA |
NA |
NA |
NA |
BindingDB |
| APP |
4-Chloro-5-(ethylsulfamoyl)-2-(furan-2-ylmethylamino)benzoic acid |
NA |
137390 |
NA |
NA |
NA |
NA |
BindingDB |
| APP |
(E)-1-(2-hydroxyethyl)-4-(2-(9-(2-(2-methoxyethoxy)ethyl)-9H-carbazol-3-yl)vinyl)pyridinium chloride |
NA |
NA |
459000 |
NA |
NA |
NA |
BindingDB |
| APP |
N-methyl-6-[2-[[6-[2-(pyridin-2-ylamino)ethyl]pyridin-2-yl]amino]ethyl]pyridin-2-amine |
NA |
280000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| APP |
6-[2-[[6-[2-(dipyridin-2-ylamino)ethyl]pyridin-2-yl]amino]ethyl]-N-methylpyridin-2-amine |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| APP |
Caffeic Acid |
NA |
NA |
NA |
216000 |
NA |
NA |
BindingDB|PubChem|TTD |
| APP |
N-Phenyl furosemide |
NA |
167530 |
NA |
NA |
NA |
NA |
BindingDB |
| APP |
4-Fluoro-2-((furan-2-ylmethyl)amino)benzoic acid |
NA |
129540 |
NA |
NA |
NA |
NA |
BindingDB |
| APP |
3-[2,5-bis(trifluoromethyl)phenyl]-N-[(1R,10S,13R)-13-[(5-chlorothiophen-2-yl)sulfonylamino]-5-tricyclo[8.2.1.03,8]trideca-3(8),4,6-trienyl]propanamide |
NA |
630000 |
NA |
NA |
NA |
NA |
BindingDB |
| APP |
US9056857, (trans)-35 |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| APP |
N-[(1R,10S,13R)-13-[(5-chlorothiophen-2-yl)sulfonylamino]-5-tricyclo[8.2.1.03,8]trideca-3(8),4,6-trienyl]-2-[[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]amino]acetamide |
NA |
800000 |
NA |
NA |
NA |
NA |
BindingDB |
| APP |
Tarenflurbil |
NA |
280000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| APP |
2-(2-Fluoro-4'-trifluoromethylbiphenyl-4-yl)propionic acid |
NA |
129000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| APP |
1-[3-Fluoro-4-[3-fluoro-4-(4-hydroxyphenyl)phenyl]phenyl]cyclopropane-1-carboxylic acid |
NA |
111000 |
NA |
NA |
NA |
NA |
BindingDB |
| AR |
N-[2-(1H-benzimidazol-2-ylsulfanyl)ethyl]aniline |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| AR |
Enzalutamide |
NA |
NA |
295400 |
NA |
NA |
NA |
BindingDB|PubChem |