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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
AR AR antagonist 3 NA NA 76000000 NA NA NA BindingDB
AR Phenol NA NA NA NA 223872 NA PubChem
ARG1 (2S)-2-amino-5-(2-aminoimidazol-1-yl)pentanoic Acid 30000000 NA NA NA NA NA BindingDB
ARG1 2-Aminohistidine 300000 NA NA NA NA NA BindingDB
ARG1 2-[4-(Diaminomethylideneamino)phenyl]-2-fluoroacetic acid 275000 NA NA NA NA NA BindingDB
ARG1 2-Acetyloxy-2-[4-(diaminomethylideneamino)phenyl]acetic acid 382000 NA NA NA NA NA BindingDB
ARG1 (2s)-2-Amino-4-(2-Amino-1h-Imidazol-5-Yl)butanoic Acid 3000000 NA NA NA NA NA BindingDB
ARG1 (S)-2-amino-5-(imidazol-2-ylamino)pentanoic acid 500000 NA NA NA NA NA BindingDB
ARG1 4-[(3,4-Dihydroxyanilino)methyl]benzene-1,2-diol NA 794000 NA NA NA NA BindingDB
ARG1 Piceatannol NA 1176000 NA NA NA NA BindingDB|PubChem
ARG1 2-Aminoimidazole 3600000 NA NA NA NA NA BindingDB
ARG2 2-[4-(Diaminomethylideneamino)phenyl]-2-fluoroacetic acid 322000 NA NA NA NA NA BindingDB|TTD
ARG2 2-Acetyloxy-2-[4-(diaminomethylideneamino)phenyl]acetic acid 437000 NA NA NA NA NA BindingDB|TTD
ARG2 (2S)-2-amino-6-borono-2-(2-piperidin-1-ylethyl)hexanoic acid NA 300000 NA NA NA NA TTD
ASAH1 Oleoyl Ethanolamide NA|500000 500000|NA NA NA NA NA PubChem
ASAH2 D-Nmappd NA 120000 NA NA NA NA BindingDB
ASAH2 12-(dimethylamino)-N-[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]dodecanamide NA 120000 NA NA NA NA BindingDB
ASGR1 D-Galactopyranose, 2-(acetylamino)-2-deoxy-, 1,3,4,6-tetraacetate NA NA|113000 150000|NA NA NA NA BindingDB|TTD
ASGR1 N-[(2S,3R,4R,5R)-4,5-dihydroxy-6,6-bis(hydroxymethyl)-2-methoxyoxan-3-yl]acetamide NA NA 199000|250000 NA NA NA BindingDB
ASGR1 (2R,3R,4S,5S,6R)-2,3,4,5-tetramethoxy-6-(methoxymethyl)tetrahydro-2H-pyran NA NA|1828000 2200000|NA NA NA NA BindingDB|TTD