GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
AR |
AR antagonist 3 |
NA |
NA |
76000000 |
NA |
NA |
NA |
BindingDB |
AR |
Phenol |
NA |
NA |
NA |
NA |
223872 |
NA |
PubChem |
ARG1 |
(2S)-2-amino-5-(2-aminoimidazol-1-yl)pentanoic Acid |
30000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ARG1 |
2-Aminohistidine |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ARG1 |
2-[4-(Diaminomethylideneamino)phenyl]-2-fluoroacetic acid |
275000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ARG1 |
2-Acetyloxy-2-[4-(diaminomethylideneamino)phenyl]acetic acid |
382000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ARG1 |
(2s)-2-Amino-4-(2-Amino-1h-Imidazol-5-Yl)butanoic Acid |
3000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ARG1 |
(S)-2-amino-5-(imidazol-2-ylamino)pentanoic acid |
500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ARG1 |
4-[(3,4-Dihydroxyanilino)methyl]benzene-1,2-diol |
NA |
794000 |
NA |
NA |
NA |
NA |
BindingDB |
ARG1 |
Piceatannol |
NA |
1176000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
ARG1 |
2-Aminoimidazole |
3600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
ARG2 |
2-[4-(Diaminomethylideneamino)phenyl]-2-fluoroacetic acid |
322000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ARG2 |
2-Acetyloxy-2-[4-(diaminomethylideneamino)phenyl]acetic acid |
437000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ARG2 |
(2S)-2-amino-6-borono-2-(2-piperidin-1-ylethyl)hexanoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
ASAH1 |
Oleoyl Ethanolamide |
NA|500000 |
500000|NA |
NA |
NA |
NA |
NA |
PubChem |
ASAH2 |
D-Nmappd |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
ASAH2 |
12-(dimethylamino)-N-[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]dodecanamide |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
ASGR1 |
D-Galactopyranose, 2-(acetylamino)-2-deoxy-, 1,3,4,6-tetraacetate |
NA |
NA|113000 |
150000|NA |
NA |
NA |
NA |
BindingDB|TTD |
ASGR1 |
N-[(2S,3R,4R,5R)-4,5-dihydroxy-6,6-bis(hydroxymethyl)-2-methoxyoxan-3-yl]acetamide |
NA |
NA |
199000|250000 |
NA |
NA |
NA |
BindingDB |
ASGR1 |
(2R,3R,4S,5S,6R)-2,3,4,5-tetramethoxy-6-(methoxymethyl)tetrahydro-2H-pyran |
NA |
NA|1828000 |
2200000|NA |
NA |
NA |
NA |
BindingDB|TTD |