GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ASGR1 |
alpha-D-Galactopyranoside, methyl 2,3,4,6-tetra-O-methyl- |
NA |
NA|2831000 |
2760000|NA |
NA |
NA |
NA |
BindingDB|TTD |
ASGR1 |
N-[(1S,2R,3R,4R,5R)-2,3-dihydroxy-1-(hydroxymethyl)-6,8-dioxabicyclo[3.2.1]octan-4-yl]methanesulfonamide |
NA |
NA |
112000 |
NA |
NA |
NA |
BindingDB |
ASGR1 |
N-[(1S,2R,3R,4R,5R)-2,3-dihydroxy-1-(hydroxymethyl)-6,8-dioxabicyclo[3.2.1]octan-4-yl]-N-methylmethanesulfonamide |
NA |
NA |
110000|161000 |
NA |
NA |
NA |
BindingDB |
ASGR1 |
beta-D-GALACTOPYRANOSE |
NA |
NA|1049000 |
1460000|NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
ASGR1 |
Glucosides |
NA |
NA|30000000 |
10000000|NA |
NA |
NA |
NA |
PubChem|TTD |
ASIC1 |
Ibuprofen |
NA |
350000 |
NA |
NA |
NA |
NA |
GtoPDB |
ASIC3 |
(3-Methoxy-pyridin-2-yl)-(6-methyl-pyridin-2-yl)-amine |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
ASIC3 |
6-Bromo-1,2,3,4-tetrahydroisoquinoline |
NA |
701000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
ASIC3 |
Agmatine |
NA |
NA |
NA |
9800000 |
NA |
NA |
GtoPDB |
ASIC3 |
Arcaine |
NA |
NA |
NA |
1200000 |
NA |
NA |
GtoPDB |
ASIC3 |
2-(3,5-dichlorophenyl)-1H-indole-5-carboximidamide |
NA |
133000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ASIC3 |
2-(3-fluoro-5-methoxyphenyl)-1H-indole-5-carboximidamide |
NA |
374000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ASIC3 |
4-(1H-Imidazol-4-YL)-benzylamine |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
ASIC3 |
Salicylic Acid |
NA |
260000 |
NA |
NA |
NA |
NA |
GtoPDB |
ASIC3 |
1-(4-Methylquinazolin-2-yl)guanidine |
NA |
NA |
NA |
1000000 |
NA |
NA |
GtoPDB |
ASIC3 |
1,3-Benzothiazol-2-ylmethylamine |
NA |
363000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
ASIC3 |
2-phenyl-1H-indole-5-carboximidamide |
NA |
2765000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ASIC3 |
2-(2,3,5-trichlorophenyl)-1H-indole-5-carboximidamide |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ASIC3 |
2-(3-chloro-5-fluorophenyl)-1H-indole-5-carboximidamide |
NA |
278000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ASIC3 |
2-(2,6-dichloropyridin-4-yl)-1H-indole-5-carboximidamide |
NA |
291000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |