GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ASIC3 |
2-(3-chloro-5-((phenylamino)methyl)phenyl)-1H-indole-5-carboximidamide |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ASIC3 |
2-(3,5-dichloro-4-cyanophenyl)-1H-indole-5-carboximidamide |
NA |
272000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ASIC3 |
2-((5-methoxy-1H-indol-3-yl)methyl)-6-(3-(trifluoromethyl)phenyl)-1,2,3,4-tetrahydroisoquinoline |
NA |
103000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
ASIC3 |
6-Phenylpyridin-2-amine |
NA |
763000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
ASIC3 |
6-Phenylpyrimidin-4-amine |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
ASIC3 |
4-(1H-imidazol-4-yl)aniline |
NA |
430000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
ATAD2 |
Thymine |
NA |
NA |
1e+07|10000000 |
NA |
NA |
NA |
ChEMBL|PubChem |
ATAD2 |
8-[2-(dimethylamino)ethylamino]-3-methyl-1H-1,7-naphthyridin-2-one |
NA |
501187|501187.23 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
ATAD2 |
N-(4-tert-butyl-1,3-thiazol-2-yl)cyclobutanecarboxamide |
NA |
NA |
500000|5e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
(2~{R})-2-azanyl-~{N}-(4-oxidanylidene-6,7-dihydro-5~{H}-1,3-benzothiazol-2-yl)propanamide |
NA |
150000 |
NA |
NA |
NA |
NA |
PubChem |
ATAD2 |
(2R)-N-(4-acetyl-1,3-thiazol-2-yl)-2-(diaminomethylideneamino)propanamide |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
ATAD2 |
1-bromo-3-[4-[(E)-2-naphthalen-1-ylethenyl]pyridin-1-ium-1-yl]propan-2-one |
NA |
822000 |
NA |
NA |
NA |
NA |
BindingDB |
ATAD2 |
ethyl 2-[3-methyl-4-[(E)-2-naphthalen-1-ylethenyl]pyridin-1-ium-1-yl]acetate |
NA |
377000 |
NA |
NA |
NA |
NA |
BindingDB |
ATAD2 |
N-(4-fluoro-3-piperidin-1-ylsulfonylphenyl)propanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
ATAD2 |
N-(4-ethyl-3-piperidin-1-ylsulfonylphenyl)propanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
ATAD2 |
N-(4-hydroxy-3-piperidin-1-ylsulfonylphenyl)propanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
ATAD2 |
N-(4-cyano-3-piperidin-1-ylsulfonylphenyl)propanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
ATAD2 |
N-(4-amino-3-piperidin-1-ylsulfonylphenyl)propanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
ATAD2 |
N-[3-piperidin-1-ylsulfonyl-4-(trifluoromethyl)phenyl]propanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
ATAD2 |
(7-amino-3,4-dihydroquinolin-1(2H)-yl)(cyclopropyl)methanone |
NA |
NA |
650000 |
NA |
NA |
NA |
BindingDB|ChEMBL |