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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ASIC3 2-(3-chloro-5-((phenylamino)methyl)phenyl)-1H-indole-5-carboximidamide NA 114000 NA NA NA NA BindingDB|TTD
ASIC3 2-(3,5-dichloro-4-cyanophenyl)-1H-indole-5-carboximidamide NA 272000 NA NA NA NA BindingDB|TTD
ASIC3 2-((5-methoxy-1H-indol-3-yl)methyl)-6-(3-(trifluoromethyl)phenyl)-1,2,3,4-tetrahydroisoquinoline NA 103000 NA NA NA NA BindingDB|TTD
ASIC3 6-Phenylpyridin-2-amine NA 763000 NA NA NA NA BindingDB|ChEMBL|TTD
ASIC3 6-Phenylpyrimidin-4-amine NA 130000 NA NA NA NA BindingDB|ChEMBL|TTD
ASIC3 4-(1H-imidazol-4-yl)aniline NA 430000 NA NA NA NA BindingDB|ChEMBL|TTD
ATAD2 Thymine NA NA 1e+07|10000000 NA NA NA ChEMBL|PubChem
ATAD2 8-[2-(dimethylamino)ethylamino]-3-methyl-1H-1,7-naphthyridin-2-one NA 501187|501187.23 NA NA NA NA BindingDB|ChEMBL|TTD
ATAD2 N-(4-tert-butyl-1,3-thiazol-2-yl)cyclobutanecarboxamide NA NA 500000|5e+05 NA NA NA BindingDB|ChEMBL
ATAD2 (2~{R})-2-azanyl-~{N}-(4-oxidanylidene-6,7-dihydro-5~{H}-1,3-benzothiazol-2-yl)propanamide NA 150000 NA NA NA NA PubChem
ATAD2 (2R)-N-(4-acetyl-1,3-thiazol-2-yl)-2-(diaminomethylideneamino)propanamide NA 140000 NA NA NA NA BindingDB
ATAD2 1-bromo-3-[4-[(E)-2-naphthalen-1-ylethenyl]pyridin-1-ium-1-yl]propan-2-one NA 822000 NA NA NA NA BindingDB
ATAD2 ethyl 2-[3-methyl-4-[(E)-2-naphthalen-1-ylethenyl]pyridin-1-ium-1-yl]acetate NA 377000 NA NA NA NA BindingDB
ATAD2 N-(4-fluoro-3-piperidin-1-ylsulfonylphenyl)propanamide NA 1000000 NA NA NA NA TTD
ATAD2 N-(4-ethyl-3-piperidin-1-ylsulfonylphenyl)propanamide NA 1000000 NA NA NA NA TTD
ATAD2 N-(4-hydroxy-3-piperidin-1-ylsulfonylphenyl)propanamide NA 1000000 NA NA NA NA TTD
ATAD2 N-(4-cyano-3-piperidin-1-ylsulfonylphenyl)propanamide NA 1000000 NA NA NA NA TTD
ATAD2 N-(4-amino-3-piperidin-1-ylsulfonylphenyl)propanamide NA 1000000 NA NA NA NA TTD
ATAD2 N-[3-piperidin-1-ylsulfonyl-4-(trifluoromethyl)phenyl]propanamide NA 1000000 NA NA NA NA TTD
ATAD2 (7-amino-3,4-dihydroquinolin-1(2H)-yl)(cyclopropyl)methanone NA NA 650000 NA NA NA BindingDB|ChEMBL