| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ATG4B |
(2E)-N-[(E)-2,3-dihydro-1H-inden-5-ylmethylideneamino]-2-(3-oxo-1,4-dihydroquinoxalin-2-ylidene)acetamide |
NA |
104000 |
NA |
NA |
NA |
NA |
BindingDB |
| ATG4B |
6-[(3-chloro-2-hydroxypropyl)amino]-1H-benzo[cd]indol-2-one |
NA |
280000 |
NA |
NA |
NA |
NA |
BindingDB |
| ATG4B |
4-[[(2S)-2-hydroxybutyl]amino]-1H-benzo[cd]indol-2-one |
NA |
113000 |
NA |
NA |
NA |
NA |
BindingDB |
| ATG4B |
4-(2-hydroxyhexylamino)-1H-benzo[cd]indol-2-one |
NA |
215000|235000 |
NA |
NA |
NA |
NA |
BindingDB |
| ATG4B |
(2E)-2-(6,7-dichloro-3-oxo-1,4-dihydroquinoxalin-2-ylidene)-N-[(E)-(2-hydroxyphenyl)methylideneamino]acetamide |
NA |
315000 |
NA |
NA |
NA |
NA |
BindingDB |
| ATG4B |
4-[(3-chloro-2-hydroxypropyl)amino]-1H-benzo[cd]indol-2-one |
NA |
132000 |
NA |
NA |
NA |
NA |
BindingDB |
| ATG4B |
(E)-4-oxo-4-(4-propylphenyl)but-2-enoic acid |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| ATG4B |
3-Benzoylacrylic acid |
NA |
580000 |
NA |
NA |
NA |
NA |
BindingDB |
| ATIC |
Pemetrexed |
200000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| ATIC |
Ddathf |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| ATIC |
2-[[4-[[(2-amino-4-oxo-3H-pyrido[2,3-d]pyrimidin-6-yl)-methylamino]methyl]benzoyl]amino]pentanedioic acid |
NA |
141000 |
NA |
NA |
NA |
NA |
TTD |
| ATIC |
|
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| ATIC |
4-(2-(3-carboxy-4-oxonaphthalen-1(4H)-ylidene)-1-phenylethyl)-1-hydroxy-2-naphthoic acid |
NA |
203700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ATIC |
[(1R,6S,10R,11S,12S,14R,22R,23S,25R)-1,10,11,12,14,23-hexahydroxy-6,10,19-trimethyl-24-oxa-4-azaheptacyclo[12.12.0.02,11.04,9.015,25.018,23.019,25]hexacosan-22-yl] 3,4-dimethoxybenzoate |
NA |
231300 |
NA |
NA |
NA |
NA |
BindingDB |
| ATIC |
Veratridine |
NA |
231300 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ATIC |
Ac-Arg-Phe-NHEt |
339000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ATIC |
Ac-Arg-Phe(4-F)-NHEt |
135000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ATIC |
Ac-Arg-N(Me)Tyr-NHEt |
145000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ATM |
Schisandrin B |
NA |
1740000 |
NA |
NA |
NA |
NA |
TTD |
| ATM |
Caffeine |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |