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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ATAD2 3,3,6-trimethyl-1H-pyrrolo[2,3-c]pyridine-2,5-dione NA NA 2400000 NA NA NA BindingDB|ChEMBL
ATAD2 Benzenamine, 3-[5-(2-thienyl)-1,3,4-oxadiazol-2-yl]- NA NA 450000 NA NA NA BindingDB|ChEMBL
ATAD2 5,6,7,8-Tetrahydrospiro[3,1-benzothiazine-4,1'-cyclohexan]-2-amine NA NA 400000|4e+05 NA NA NA BindingDB|ChEMBL
ATAD2 N-[4-methoxy-3-(piperidin-1-ylsulfonyl)phenyl]propanamide NA 1000000 NA NA NA NA TTD
ATAD2 3-Methyl-1,5-naphthyridin-2-ol NA NA 600000|6e+05 NA NA NA BindingDB|ChEMBL
ATAD2 3-(5-Phenyl-4h-1,2,4-Triazol-3-Yl)aniline NA NA 350000 NA NA NA BindingDB|ChEMBL
ATAD2 6-Amino-1-ethyl-1,2,3,4-tetrahydroquinolin-2-one NA NA 650000 NA NA NA BindingDB|ChEMBL
ATAD2 3-methylquinolin-2(1H)-one NA 1000000 NA NA NA NA TTD
ATAD2 3-[4-[(E)-2-naphthalen-1-ylethenyl]pyridin-1-ium-1-yl]propan-1-amine NA 543000 NA NA NA NA BindingDB
ATAD2 Thymidine NA NA 1e+07|10000000 NA NA NA ChEMBL|PubChem
ATAD2 2-Amino-7,7-dimethyl-5,6,7,8-tetrahydro-4H-[1,3]thiazolo[5,4-c]azepin-4-one NA NA 500000|5e+05 NA NA NA BindingDB|ChEMBL
ATAD2 (2R)-N-(4-acetyl-1,3-thiazol-2-yl)-2-aminopropanamide NA 336000 NA NA NA NA BindingDB
ATAD2 2-(5-Pyridin-4-yl-1,3,4-oxadiazol-2-yl)aniline NA NA 600000|6e+05 NA NA NA BindingDB|ChEMBL
ATAD2 5-amino-1,3,6-trimethyl-1,3-dihydro-2H-benzimidazol-2-one NA NA 600000|6e+05 NA NA NA BindingDB|ChEMBL
ATAD2 4-(5-Phenyl-1,3,4-oxadiazol-2-yl)pyridine NA NA 400000|4e+05 NA NA NA BindingDB|ChEMBL
ATAD2 N-(6-methoxy-1,3-benzothiazol-2-yl)-2-methylpropanamide NA NA 450000 NA NA NA BindingDB|ChEMBL
ATAD2 Methyl 3-Amino-5-(3,5-Dimethyl-1,2-Oxazol-4-Yl)benzoate NA NA 2e+05 NA NA NA ChEMBL
ATG4B 4-(1H-perimidin-2-yl)phenol NA 150000|300000 NA NA NA NA BindingDB
ATG4B 4-[[(2R)-2-hydroxybutyl]amino]-1H-benzo[cd]indol-2-one NA 119000 NA NA NA NA BindingDB
ATG4B 4-(2-hydroxybutylamino)-1H-benzo[cd]indol-2-one NA 111000 NA NA NA NA BindingDB