GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ATAD2 |
3,3,6-trimethyl-1H-pyrrolo[2,3-c]pyridine-2,5-dione |
NA |
NA |
2400000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
Benzenamine, 3-[5-(2-thienyl)-1,3,4-oxadiazol-2-yl]- |
NA |
NA |
450000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
5,6,7,8-Tetrahydrospiro[3,1-benzothiazine-4,1'-cyclohexan]-2-amine |
NA |
NA |
400000|4e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
N-[4-methoxy-3-(piperidin-1-ylsulfonyl)phenyl]propanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
ATAD2 |
3-Methyl-1,5-naphthyridin-2-ol |
NA |
NA |
600000|6e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
3-(5-Phenyl-4h-1,2,4-Triazol-3-Yl)aniline |
NA |
NA |
350000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
6-Amino-1-ethyl-1,2,3,4-tetrahydroquinolin-2-one |
NA |
NA |
650000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
3-methylquinolin-2(1H)-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
ATAD2 |
3-[4-[(E)-2-naphthalen-1-ylethenyl]pyridin-1-ium-1-yl]propan-1-amine |
NA |
543000 |
NA |
NA |
NA |
NA |
BindingDB |
ATAD2 |
Thymidine |
NA |
NA |
1e+07|10000000 |
NA |
NA |
NA |
ChEMBL|PubChem |
ATAD2 |
2-Amino-7,7-dimethyl-5,6,7,8-tetrahydro-4H-[1,3]thiazolo[5,4-c]azepin-4-one |
NA |
NA |
500000|5e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
(2R)-N-(4-acetyl-1,3-thiazol-2-yl)-2-aminopropanamide |
NA |
336000 |
NA |
NA |
NA |
NA |
BindingDB |
ATAD2 |
2-(5-Pyridin-4-yl-1,3,4-oxadiazol-2-yl)aniline |
NA |
NA |
600000|6e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
5-amino-1,3,6-trimethyl-1,3-dihydro-2H-benzimidazol-2-one |
NA |
NA |
600000|6e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
4-(5-Phenyl-1,3,4-oxadiazol-2-yl)pyridine |
NA |
NA |
400000|4e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
N-(6-methoxy-1,3-benzothiazol-2-yl)-2-methylpropanamide |
NA |
NA |
450000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
ATAD2 |
Methyl 3-Amino-5-(3,5-Dimethyl-1,2-Oxazol-4-Yl)benzoate |
NA |
NA |
2e+05 |
NA |
NA |
NA |
ChEMBL |
ATG4B |
4-(1H-perimidin-2-yl)phenol |
NA |
150000|300000 |
NA |
NA |
NA |
NA |
BindingDB |
ATG4B |
4-[[(2R)-2-hydroxybutyl]amino]-1H-benzo[cd]indol-2-one |
NA |
119000 |
NA |
NA |
NA |
NA |
BindingDB |
ATG4B |
4-(2-hydroxybutylamino)-1H-benzo[cd]indol-2-one |
NA |
111000 |
NA |
NA |
NA |
NA |
BindingDB |