| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ATP4A |
2-(5,6-Dimethoxy-1H-benzoimidazole-2-sulfinylmethyl)-phenylamine |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ATP4A |
[2-Methyl-8-(3-phenyl-allyl)-imidazo[1,2-a]pyridin-3-yl]-acetonitrile |
NA |
206000|442000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ATP4A |
Timoprazole |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ATP4B |
2-(5,6-Dimethoxy-1H-benzoimidazole-2-sulfinylmethyl)-phenylamine |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| ATP4B |
[2-Methyl-8-(3-phenyl-allyl)-imidazo[1,2-a]pyridin-3-yl]-acetonitrile |
NA |
442000 |
NA |
NA |
NA |
NA |
TTD |
| ATP4B |
Timoprazole |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| ATR |
Caffeine |
NA |
1100000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| ATXN2 |
Ouabain |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| ATXN2 |
Digitoxin |
NA |
NA |
NA |
NA |
501187 |
NA |
PubChem |
| AURKA |
5-Amino-[3,3'-bipyridin]-6(1H)-one |
125200 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| AURKA |
3-(1H-benzimidazol-2-yl)-6-chloro-1H-benzimidazol-2-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| AURKA |
(5Z)-3-(cyclohexylmethyl)-2-(4-ethylphenyl)imino-5-(pyridin-4-ylmethylidene)-1,3-thiazolidin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| AURKA |
[3,4'-Bipyridin]-5-amine, 6-methoxy- |
184700 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| AURKA |
5-(1-hydroxynaphthalen-2-yl)-N-(3-methoxyphenyl)-3-(4-methoxyphenyl)-3,4-dihydropyrazole-2-carbothioamide |
NA |
105030 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| AURKA |
1-O-[[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl] 4-O-[(3R)-3-hydroxy-2,2-dimethyl-4-oxo-4-[[3-oxo-3-(2-sulfanylethylamino)propyl]amino]butyl] butanedioate |
NA |
117000|731000 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKA |
1-O-[[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl] 5-O-[(3R)-3-hydroxy-2,2-dimethyl-4-oxo-4-[[3-oxo-3-(propylamino)propyl]amino]butyl] pentanedioate |
NA |
542000 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKA |
1-O-[[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl] 4-O-[(3R)-3-hydroxy-2,2-dimethyl-4-oxo-4-[[3-oxo-3-(propylamino)propyl]amino]butyl] butanedioate |
NA |
497000 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKA |
1-O-[[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl] 4-O-[(3R)-3-hydroxy-2,2-dimethyl-4-(methylamino)-4-oxobutyl] butanedioate |
NA |
1300000 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKA |
[[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(3S)-4-[[3-(ethylamino)-3-oxopropyl]amino]-3-hydroxy-2,2-dimethyl-4-oxobutyl] hydrogen phosphate |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKA |
1-O-[[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl] 4-O-[(3R)-3-hydroxy-2,2-dimethyl-4-[[3-(methylamino)-3-oxopropyl]amino]-4-oxobutyl] butanedioate |
NA |
1400000 |
NA |
NA |
NA |
NA |
BindingDB |