| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| AURKA |
Kinase inhibitor, A2 |
NA |
188000 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKB |
5-amino-1-methyl-[3,4'-bipyridin]-6(1H)-one |
102700 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| AURKB |
N-cyclohexyl-6-(1H-indazol-5-yl)imidazo[2,1-b]thiazol-5-amine |
1800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| AURKB |
3-Amino-2-pyridinol |
159700 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| AURKB |
(S)-3-Hydroxy Midostaurin |
NA |
NA |
750000 |
NA |
NA |
NA |
BindingDB |
| AURKB |
4-Chloro-3-(pyridin-2-ylmethoxy)aniline |
NA |
125893 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKC |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AVPR1A |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| AVPR1A |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| AVPR1A |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| AVPR1A |
5-(2,3-dimethylphenyl)-N-(2-methoxyethyl)-N-(6-methoxypyridin-3-yl)pyrazine-2-carboxamide |
539000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AVPR1A |
5-(2,3-dimethylphenyl)-N-ethyl-N-(6-methoxypyridin-3-yl)pyrazine-2-carboxamide |
472000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AVPR1A |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| AVPR1A |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| AVPR1A |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| AVPR1A |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| AVPR1A |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| AVPR2 |
(10R,13S,16S,19S)-N-[(2S)-1-[[(2R)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-19-(2-amino-2-oxoethyl)-13-benzyl-10-[(4-ethoxyphenyl)methyl]-8,11,14,17,20-pentaoxo-16-propan-2-yl-9,12,15,18,21-pentazaspiro[5.19]pentacosane-22-carboxamide |
400000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AVPR2 |
N-ethyl-5-(3-fluoro-2-methylphenyl)-N-(6-methoxypyridin-3-yl)pyrazine-2-carboxamide |
343000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AVPR2 |
(13S,16S,19S,22R)-N-[(2S)-1-[[(2R)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-13-(2-amino-2-oxoethyl)-19-benzyl-22-[(4-ethoxyphenyl)methyl]-12,15,18,21,24-pentaoxo-16-propan-2-yl-7,8-dithia-11,14,17,20,23-pentazaspiro[5.19]pentacosane-10-carboxamide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |