| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| AURKA |
3-[[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methylamino]-3-oxopropanoic acid |
NA |
910000 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKA |
1-O-[[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl] 3-O-[(3R)-3-hydroxy-2,2-dimethyl-4-oxo-4-[[3-oxo-3-(propylamino)propyl]amino]butyl] propanedioate |
NA |
1300000 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKA |
1-O-[[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl] 4-O-(2,2-dimethylpropyl) butanedioate |
NA |
430000 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKA |
[(3R)-3-hydroxy-2,2-dimethyl-4-oxo-4-[[3-oxo-3-(propylamino)propyl]amino]butyl] 3-[[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methylamino]-3-oxopropanoate |
NA |
1100000 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKA |
3-[[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy]-3-oxopropanoic acid |
NA |
420000 |
NA |
NA |
NA |
NA |
BindingDB |
| AURKA |
3-Amino-2-pyridinol |
361000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| AURKA |
Amrinone |
393900 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|PubChem|TTD |
| AURKA |
AR-AO-14418 |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| AURKA |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AURKA |
1-[(4-methoxyphenyl)methyl]-3-[6-(2H-tetrazol-5-yl)-1,3-benzothiazol-2-yl]urea |
NA |
4800000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| AURKA |
1-[(4-methoxyphenyl)methyl]-3-[4-(2H-tetrazol-5-yl)pyridin-2-yl]urea |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| AURKA |
N-[3-[3-[[2-methyl-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]amino]-1H-pyrazol-5-yl]phenyl]butane-1-sulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| AURKA |
1-[(4-Methoxyphenyl)methyl]-3-(6-nitro-1,3-benzothiazol-2-yl)urea |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| AURKA |
1-(4-Cyanopyridin-2-yl)-3-[(4-methoxyphenyl)methyl]urea |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| AURKA |
N-[3-[3-[[2-methyl-6-(2-morpholin-4-ylethylamino)pyrimidin-4-yl]amino]-1H-pyrazol-5-yl]phenyl]benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| AURKA |
3-methyl-N-[3-[3-[[2-methyl-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]amino]-1H-pyrazol-5-yl]phenyl]benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| AURKA |
N-[3-[3-[[6-[2-(dimethylamino)ethylamino]-2-methylpyrimidin-4-yl]amino]-1H-pyrazol-5-yl]phenyl]benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| AURKA |
H-Cys(1)-Asp-Gly-Val-Pro-Trp-His-Cys(1)-Gly-NH2 |
NA |
242000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| AURKA |
H-Cys(1)-His-Pro-Gln-Gly-Asp-Thr-Cys(1)-Gly-NH2 |
NA |
137000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| AURKA |
H-Cys(1)-Gly-His-Pro-Gln-Val-Pro-Cys(1)-Gly-NH2 |
NA |
234000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |