| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| AVPR2 |
(2R)-N-[(2S)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-1-[(13S,16S,19S,22R)-13-(2-amino-2-oxoethyl)-19-benzyl-22-[(4-ethoxyphenyl)methyl]-12,15,18,21,24-pentaoxo-16-propan-2-yl-7,8-dithia-11,14,17,20,23-pentazaspiro[5.19]pentacosane-10-carbonyl]pyrrolidine-2-carboxamide |
1100000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AVPR2 |
(2R)-N-[(2S)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-1-[(10R,13S,16S,19S)-19-(2-amino-2-oxoethyl)-13-benzyl-10-[(4-ethoxyphenyl)methyl]-8,11,14,17,20-pentaoxo-16-propan-2-yl-9,12,15,18,21-pentazaspiro[5.19]pentacosane-22-carbonyl]pyrrolidine-2-carboxamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AVPR2 |
(13S,16S,19S,22R)-N-[(2S)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-13-(2-amino-2-oxoethyl)-19-benzyl-22-[(4-ethoxyphenyl)methyl]-12,15,18,21,24-pentaoxo-16-propan-2-yl-7,8-dithia-11,14,17,20,23-pentazaspiro[5.19]pentacosane-10-carboxamide |
1500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| AXL |
4-Chloro-1H-pyrrolo[2,3-b]pyridine |
NA |
113000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
3-Bromopyrazolo(1,5-a)pyrimidine |
NA |
330000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
5-Bromo-6-methoxy-1H-indazole |
NA |
227000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
N-(1-methylpiperidin-4-yl)-3-(1-methylpyrazol-4-yl)-1H-indazol-5-amine |
NA |
207000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
N-[(1-methylpiperidin-4-yl)methyl]-3-(1-methylpyrazol-4-yl)-1H-indazol-5-amine |
NA |
1850000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
N-methyl-1-[3-(1-methylpyrazol-4-yl)-1H-indazol-5-yl]pyrrolidin-3-amine |
NA |
432000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
3-(1-methylpyrazol-4-yl)-N-[(3S)-pyrrolidin-3-yl]-1H-indazol-5-amine |
NA |
239000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
3-(1-methylpyrazol-4-yl)-N-pyrrolidin-3-yl-1H-indazol-5-amine |
NA |
132000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
3-(1-methylpyrazol-4-yl)-N-phenyl-1H-indazol-6-amine |
NA |
219000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
4-bromo-1H-indazole |
NA |
178000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
3-Bromo-1H-indazol-4-amine |
NA |
486000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
4-(Trifluoromethyl)-1H-indazole |
NA |
184000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
2,4-Di(3-pyridyl)-1,3-thiazole |
NA |
305000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
4-Chlorothieno[3,2-d]pyrimidine |
NA |
302000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
5-(4-Fluorophenyl)-3-(methylsulfanyl)-1H-pyrazole |
NA |
331000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
6-Methyl-4-(piperazin-1-yl)-2-(trifluoromethyl)quinoline |
NA |
204000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
2-Amino-6-fluorobenzothiazole |
NA |
363000 |
NA |
NA |
NA |
NA |
ChEMBL |