| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| AXL |
3-(Pyridin-3-yl)aniline |
NA |
363000 |
NA |
NA |
NA |
NA |
ChEMBL |
| AXL |
1H-Pyrrolo(2,3-b)pyridine |
NA |
391000 |
NA |
NA |
NA |
NA |
ChEMBL |
| B2M |
(4S,4aS,5aS,6S,12aS)-4-(dimethylamino)-6,10,12a-trihydroxy-6-methyl-1,3,11,12-tetraoxo-N-(pyrrolidin-1-ylmethyl)-4a,5,5a,11a-tetrahydro-4H-tetracene-2-carboxamide |
NA |
136000 |
NA |
NA |
NA |
NA |
BindingDB |
| B2M |
(4S,4aS,12aR)-7-chloro-4-(dimethylamino)-10,11,12a-trihydroxy-6-methyl-1,3,12-trioxo-4a,5-dihydro-4H-tetracene-2-carboxamide |
NA |
136000 |
NA |
NA |
NA |
NA |
BindingDB |
| B3GALT1 |
1-Methyl-3-[20-(3-methylimidazol-3-ium-1-yl)icosyl]imidazol-1-ium |
NA |
420000|440000 |
NA |
NA |
NA |
NA |
BindingDB |
| B3GALT1 |
1-Methyl-3-[22-(3-methylimidazol-3-ium-1-yl)docosyl]imidazol-1-ium |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB |
| B4GALT1 |
1-Methyl-3-[20-(3-methylimidazol-3-ium-1-yl)icosyl]imidazol-1-ium |
NA |
1960000 |
NA |
NA |
NA |
NA |
BindingDB |
| B4GALT1 |
[[(2R,3S,4R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4S,5R,6S)-3,4,5-trihydroxy-6-[2-[2-(2-methoxyethoxy)ethoxy]ethoxymethyl]oxan-2-yl] hydrogen phosphate |
149000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
4,9-Bis[(3-methylbut-2-en-1-yl)oxy]-7H-furo[3,2-g]chromen-7-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
Byakangelicin |
NA |
219700 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
(4S)-4-amino-5-[[(2S,3S)-1-[[(2S)-1-[[(2R,3S,4S)-3-hydroxy-6-methyl-2-(4-methylanilino)heptan-4-yl]amino]-1-oxo-3-thiophen-2-ylpropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-5-oxopentanoic acid |
NA |
813000 |
NA |
NA |
NA |
NA |
BindingDB |
| BACE1 |
Osthol |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| BACE1 |
Ninhydrin |
NA |
776000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
4a,5,6,7,8,8a-hexahydro-4H-3,1-benzothiazin-2-amine |
NA |
4000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
N~3~-Benzylpyridine-2,3-diamine |
NA |
310000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| BACE1 |
Dihydroxanthyletin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
Angelicin |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| BACE1 |
7-Methoxycoumarin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| BACE1 |
5-{2-[3-Hydroxy-4-(2-hydroxy-2-naphthalen-1-yl-acetylamino)-6-methyl-heptanoylamino]-3-methyl-butyrylamino}-cyclohexane-1,3-dicarboxylic acid dimethyl ester |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BACE1 |
4-(Trifluoromethyl)quinolin-2-amine |
NA |
NA |
2900000 |
NA |
NA |
NA |
BindingDB |