| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCHE |
2,2'-[1,4-Phenylenebis(methylene)]di(isoquinolin-2-ium) dibromide |
NA |
840000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
1,10-Bis(isoquinolinium)-1,4-phenyldimethylenyl dibromide |
NA |
840000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
4-(5-{4-[Dimethyl(prop-2-enyl)ammonio]phenyl}-3-oxopentyl)-N,N-dimethyl-N-prop-2-enylbenzenaminium |
NA |
255000|354000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
8-Methoxy-2-(2-methylphenyl)-3,4-dihydroisoquinolin-2-ium;bromide |
NA |
133000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(2-Fluoro-4-iodophenyl)-8-methoxy-3,4-dihydroisoquinolin-2-ium;bromide |
NA |
128000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(4-Fluorophenyl)-8-methoxy-3,4-dihydroisoquinolin-2-ium;bromide |
NA |
113000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
11,13,15-Triphenyl-17-oxa-2,14,15-triazatetracyclo[8.7.0.03,8.012,16]heptadeca-1,3(8),9,12(16),13-pentaen-9-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
3-(8-Methoxy-3,4-dihydroisoquinolin-2-ium-2-yl)benzonitrile;bromide |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
8-Methoxy-2-(4-methoxyphenyl)-3,4-dihydroisoquinolin-2-ium;bromide |
NA |
113000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
8-Methoxy-2-[4-(trifluoromethyl)phenyl]-3,4-dihydroisoquinolin-2-ium;bromide |
NA |
221000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(2-Chlorophenyl)-8-methoxy-3,4-dihydroisoquinolin-2-ium;bromide |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(2,6-Difluorophenyl)-8-methoxy-3,4-dihydroisoquinolin-2-ium;bromide |
NA |
105000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(2,4-Dibromophenyl)-8-methoxy-3,4-dihydroisoquinolin-2-ium;bromide |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
Boldione |
NA |
102660 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2,2-Dimethyl-3-[methyl(methylsulfanyl)phosphoryl]oxybutane |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
Pralidoxime Iodide |
390000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
Pegamine |
NA |
105100 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(Isoquinolin-2-ium-2-ylmethyl)isoquinolin-2-ium;dibromide |
NA |
1400000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
1,1'-(Pentane-1,5-diyl)di(pyridin-1-ium) dibromide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
2-[(2-hydroxyphenyl)methylene]-N-(4-pyridinyl)-1-hydrazinecarboxamide |
212400 |
NA |
NA |
NA |
NA |
NA |
TTD |