| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCHE |
1-[(E)-4-[3-fluoro-4-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]but-2-enyl]pyridin-1-ium-4-carboxamide;dibromide |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
4-[3-[(1S)-1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-3H-2-benzofuran-5-yl]-1H-1,2,4-triazol-5-yl]phenol |
NA |
140220 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
2-[3-[(1S)-1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-3H-2-benzofuran-5-yl]-1H-1,2,4-triazol-5-yl]phenol |
NA |
101520 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
1-[(E)-(4-hydroxy-3-methoxyphenyl)methylideneamino]-3-pyridin-4-ylurea |
446480 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
1-(4-cyanophenyl)-3-[(E)-(6-hydroxy-2,4-dioxo-1H-pyrimidin-5-yl)methylideneamino]thiourea |
NA |
231000|231610 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
N-[(6-hydroxy-2,4-dioxo-1H-pyrimidin-5-yl)methylidene]acetamide |
NA |
116000|116610 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[(E)-(6-hydroxy-2,4-dioxo-1H-pyrimidin-5-yl)methylideneamino]-3-[3-(trifluoromethyl)phenyl]thiourea |
NA |
136000|136910 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
ethyl (E)-3-[3-methoxy-4-(6-pyrrolidin-1-ylhexoxy)phenyl]prop-2-enoate |
NA |
376000|376710 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
(E)-3-[4-[8-(diethylamino)octoxy]-3-methoxyphenyl]prop-2-enoic acid |
NA |
302000|302450 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
(E)-3-[3-methoxy-4-(6-pyrrolidin-1-ylhexoxy)phenyl]prop-2-enoic acid |
NA |
286000|286720 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
[(1R,3S)-3-(4-methoxyanilino)cyclohexyl] N,N-dimethylcarbamate |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
(E)-3-[3-methoxy-4-(6-piperidin-1-ylhexoxy)phenyl]prop-2-enoic acid |
NA |
145000|145690 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
[(1R,3R)-3-(4-methoxyanilino)cyclohexyl] N,N-dimethylcarbamate |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
(E)-3-[4-[6-(diethylamino)hexoxy]-3-methoxyphenyl]prop-2-enoic acid |
NA |
263000|263110 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
(E)-3-(4-Hydroxy-3-methoxyphenyl)-N-phenylacrylamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
Ganoderol B |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
Lucidenic Acid A |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
N-[dichlorophosphinyl]-4-methylbenzamide |
NA |
1200000 |
8900000 |
NA |
NA |
NA |
BindingDB |
| BCHE |
10-Benzyl-3,4,9,10,11,12-hexahydro-2H-pyrido[4',3':4,5]thieno[3,2-e]pyrimido[1,2-c]pyrimidin (14) |
NA |
119000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
5-amino-4-[4-(dimethylamino)phenyl]-3,4,6,7,8,9-hexahydro-1H-pyrimido[4,5-b]quinoline-2-thione |
NA |
154000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |