| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCHE |
1-[(E)-4-[3,5-dichloro-4-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]but-2-enyl]pyridin-1-ium-4-carboxamide;dibromide |
187000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[3-[3,5-dichloro-4-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]propyl]pyridin-1-ium-4-carboxamide;dibromide |
195000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[3-[3-chloro-4-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]propyl]pyridin-1-ium-4-carboxamide;dibromide |
273000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[(E)-4-[3-chloro-4-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]but-2-enyl]pyridin-1-ium-4-carboxamide;dibromide |
294000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[4-[3-chloro-4-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]butyl]pyridin-1-ium-4-carboxamide;dibromide |
265000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[4-[3,5-dichloro-4-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]butyl]pyridin-1-ium-4-carboxamide;dibromide |
140000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-(4-Methoxybenzyl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
[Methyl(methylsulfanyl)phosphoryl]oxycyclohexane |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-(4-nitrophenyl)-4-phenyl-1H-1,2,3-triazole |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
4-[[1-[(4-chlorophenyl)methyl]piperidin-4-yl]methoxy]-2-[2-(cyclopropanecarbonylamino)pyridin-4-yl]-N-methyl-1,3-thiazole-5-carboxamide |
NA |
297000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
1,1''-Bis(pyridinium)-1,4-phenyldimethylene dibromide |
NA |
529000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
N-(pyridin-4-yl)hydrazinecarboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
[4-[3-[Benzyl(methyl)amino]propoxy]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
(2,2-Dimethyl-8-oxo-3,4-dihydropyrano[3,2-g]chromen-3-yl) 4-[[5-(dithiolan-3-yl)pentanoylamino]methyl]triazole-1-carboxylate |
NA |
5890000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
[4-[4-[Benzyl(methyl)amino]butoxy]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone |
NA |
219000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
5',8-dichloro-1'-methylspiro[6H-pyrazolo[1,5-c]quinazoline-5,3'-indole]-2'-one |
NA |
219300 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
4-[2-[1-[(2-Chlorophenyl)methyl]piperidin-4-yl]ethoxy]-2-[2-(cyclopropanecarbonylamino)pyridin-4-yl]-1,3-thiazole-5-carboxamide |
NA |
301300 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
Dehydrodiscretamine |
NA |
118800 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
(1R,9S,10R)-16-methyl-6,14-diazatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,16-trien-5-one |
NA |
169000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
Testololactone |
NA |
142450 |
NA |
NA |
NA |
NA |
BindingDB |