| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCHE |
(-)-Corydalmine |
NA |
123600 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(4-Bromo-2-fluorophenyl)-8-methoxyisoquinolin-2-ium;bromide |
NA |
196000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(4-Chlorophenyl)-8-methoxyisoquinolin-2-ium;bromide |
NA |
104000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(2,4-Dichlorophenyl)-8-methoxyisoquinolin-2-ium;bromide |
NA |
232000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(2,4-Dibromophenyl)-8-methoxyisoquinolin-2-ium;bromide |
NA |
131000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-[2-(Cyclopropanecarbonylamino)pyridin-4-yl]-4-[2-[1-[(3-fluorophenyl)methyl]piperidin-4-yl]ethoxy]-1,3-thiazole-5-carboxamide |
NA |
294700 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(4-Bromophenyl)isoquinolin-2-ium;bromide |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(4-Fluorophenyl)-8-methoxyisoquinolin-2-ium;bromide |
NA |
143000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
8-Methoxy-2-(2-methylphenyl)isoquinolin-2-ium;bromide |
NA |
243000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
(12R)-7,16-dimethoxy-3,5-dioxa-11-azapentacyclo[10.7.1.02,6.08,20.014,19]icosa-1,6,8(20),14(19),15,17-hexaen-18-ol |
NA |
140700 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
1,1''-Bis(pyridinium)-1,2-phenyldimethylene dibromide |
NA |
345000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
N-((4-aminophenyl)sulfonyl)-2-(4-isobutylphenyl)propanamide |
NA |
214000|214410 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-(4-Chlorophenyl)-4-phenyl-1H-1,2,3-triazole |
NA |
555500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[3-[3,5-difluoro-4-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]propyl]pyridin-1-ium-4-carboxamide;dibromide |
279000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
1-[3-[3-fluoro-4-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]propyl]pyridin-1-ium-4-carboxamide;dibromide |
484000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
1-[4-[3,5-difluoro-4-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]butyl]pyridin-1-ium-4-carboxamide;dibromide |
284000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
1-[(E)-4-[3,5-difluoro-4-[(E)-hydroxyiminomethyl]pyridin-1-ium-1-yl]but-2-enyl]pyridin-1-ium-4-carboxamide;dibromide |
243000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(4-Methoxyphenyl)-9-methylpyrido[3,4-b]indol-2-ium |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
9-Methyl-2-(4-methylphenyl)pyrido[3,4-b]indol-2-ium |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(4-Chlorophenyl)-9-methylpyrido[3,4-b]indol-2-ium |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB |