| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CACNA1B |
2-[3-[4-[[[6-(4-Hydroxyphenoxy)-1,3-benzothiazol-2-yl]amino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
253000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
N-[[4-(3-aminopropoxy)phenyl]methyl]-N-methyl-6-[4-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid |
NA |
283000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
2,2,2-Trifluoroacetic acid;2-[3-[4-[[[6-[4-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-yl]amino]methyl]phenoxy]propyl]guanidine |
NA |
167000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
2-[3-[4-[[[6-(4-Cyanophenoxy)-1,3-benzothiazol-2-yl]-methylamino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
143000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
2-[3-[4-[[Methyl-[6-[4-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-yl]amino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
185000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
N-[[4-(3-aminopropoxy)phenyl]methyl]-6-(4-fluorophenoxy)-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid |
NA |
106000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
N-[[4-(3-aminopropoxy)phenyl]methyl]-6-[3-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid |
NA |
144000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
4-[[2-[[4-(3-Aminopropoxy)phenyl]methyl-methylamino]-1,3-benzothiazol-6-yl]oxy]phenol;2,2,2-trifluoroacetic acid |
NA |
117000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
2-[3-[4-[[Methyl-(6-phenoxy-1,3-benzothiazol-2-yl)amino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
113000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
N-[[4-(3-aminopropoxy)phenyl]methyl]-6-phenoxy-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid |
NA |
218000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
2-[3-[4-[[[6-(4-Cyanophenoxy)-1,3-benzothiazol-2-yl]amino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
368000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
4-[3-(dimethylamino)propoxy]-N-[2-(4-fluorophenoxy)phenyl]benzamide |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB |
| CACNA1B |
Bohemine |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CACNA1B |
Indirubin-3'-monoxime |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CACNA1B |
N-[(2S)-1-[4-[4-(1H-imidazol-5-ylmethylamino)-N-(3-methylbutyl)anilino]piperidin-1-yl]-4-methyl-1-oxopentan-2-yl]azepane-1-carboxamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1B |
Olomoucine |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CACNA1B |
Iso-Olomoucine |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CACNA1B |
(2R)-2-({6-[benzyl(methyl)amino]-9-isopropyl-9H-purin-2-yl}amino)butan-1-ol |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CACNA1B |
(S)-Seliciclib |
NA |
NA |
NA |
570000 |
NA |
NA |
TTD |
| CACNA1B |
N9-Isopropylolomoucine |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |