Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CACNA1B | Olomoucine, Dimethylamino- | NA | NA | NA | 1000000 | NA | NA | TTD |
| CACNA1B | (2R)-2-[[6-(dibenzylamino)-9-propan-2-ylpurin-2-yl]amino]butan-1-ol | NA | NA | NA | 1000000 | NA | NA | TTD |
| CACNA1B | 8-Bromo-5H-indolo[3,2-c]quinolin-6(11H)-one | NA | NA | NA | 1000000 | NA | NA | TTD |
| CACNA1C | Tadalafil | NA | 398107|398107.17 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Paliperidone | NA | 193900|398107|1000000|398107.17 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Vardenafil | NA | 251189 | NA | NA | NA | NA | PubChem |
| CACNA1C | Moxifloxacin | NA | 168900|173000|398107 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | Telbivudine | NA | 713900 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | Phenytoin | NA | 125000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Lapatinib | NA | 1995262|15848932|15848900|1995260|1995262.31 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Alfuzosin | NA | 199526|199526.23 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Darunavir | NA | 1584893|1584890|1584893.19 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Deferasirox | NA | 1000000 | NA | NA | NA | NA | PubChem|TTD |
| CACNA1C | Dasatinib | NA | 251189|398107|251188.64 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Disopyramide | NA | 1036700 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | Carticaine | NA | 471000 | NA | NA | NA | NA | PubChem |
| CACNA1C | Eugenol | NA | 187000 | NA | NA | NA | NA | PubChem |
| CACNA1C | Halothane | NA | 1800000|14500000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Ribavirin | NA | 622500 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | Isobutylmethylxanthine | NA | 466000 | NA | NA | NA | NA | BindingDB|TTD |