Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CACNA1C | Lamotrigine | NA | 1258925|1584893|1258930|1584890|1258925.41 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Metronidazole | NA | 177900 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | Piperacillin | NA | 1226000 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | Sitagliptin | NA | 147100|100000000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Linezolid | NA | 105400 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | Darifenacin | NA | 1584893|1584890|1584893.19 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | 2-[2-ethoxy-5-(4-ethylpiperazin-1-yl)sulfonylphenyl]-5-methyl-7-propyl-2,3-dihydro-1H-imidazo[5,1-f][1,2,4]triazin-4-one | NA | 251189 | NA | NA | NA | NA | BindingDB |
| CACNA1C | 6-((((1R,4r)-4-((R)-1-Amino-2-(7-methoxy-2-oxo-1,5-naphthyridin-1(2H)-yl)ethyl)cyclohexyl)amino)methyl)-2H-pyrido[3,2-b][1,4]oxazin-3(4H)-one | NA | 333000 | NA | NA | NA | NA | TTD |
| CACNA1C | 2-[[[4-[(1R)-1-amino-2-(7-fluoro-2-oxoquinoxalin-1-yl)ethyl]cyclohexyl]amino]methyl]-8H-pyrimido[5,4-b][1,4]oxazin-7-one | NA | 333000 | NA | NA | NA | NA | TTD |
| CACNA1C | Pentobarbital | NA | 299000 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | Procainamide | NA | 389500 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | Risperidone | NA | 125000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Sotalol | NA | 193300|1023000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Silodosin | NA | 794328|794328.23 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Sunitinib | NA | 199526|199526.23 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CACNA1C | Raltegravir | NA | 246700 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | Ceftriaxone | NA | 153800 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | Ranolazine | NA | 311000 | NA | NA | NA | NA | PubChem |
| CACNA1C | Mibefradil | NA | 108000|288000 | NA | NA | NA | NA | BindingDB|PubChem |
| CACNA1C | NA | 1000000 | NA | NA | NA | NA | BindingDB |