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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CACNA1D Voriconazole NA 414200 NA NA NA NA PubChem
CACNA1F Paliperidone NA 193900 NA NA NA NA PubChem
CACNA1F Moxifloxacin NA 173000 NA NA NA NA PubChem
CACNA1F Telbivudine NA 713900 NA NA NA NA PubChem
CACNA1F Disopyramide NA 1036700 NA NA NA NA PubChem
CACNA1F Ribavirin NA 622500 NA NA NA NA PubChem
CACNA1F Metronidazole NA 177900 NA NA NA NA PubChem
CACNA1F Piperacillin NA 1226000 NA NA NA NA PubChem
CACNA1F Sitagliptin NA 147100 NA NA NA NA PubChem
CACNA1F Linezolid NA 105400 NA NA NA NA PubChem
CACNA1F Pentobarbital NA 299000 NA NA NA NA PubChem
CACNA1F Procainamide NA 389500 NA NA NA NA PubChem
CACNA1F Sotalol NA 193300 NA NA NA NA PubChem
CACNA1F Raltegravir NA 246700 NA NA NA NA PubChem
CACNA1F Ceftriaxone NA 153800 NA NA NA NA PubChem
CACNA1F Voriconazole NA 414200 NA NA NA NA PubChem
CACNA1G 2-[2-[5-(dimethylamino)pentylsulfanyl]-3-phenyl-4H-quinazolin-4-yl]-N-[(4-fluorophenyl)methyl]acetamide NA 554900 NA NA NA NA BindingDB
CACNA1G N-((4-phenyl-2-propyloxazol-5-yl)methyl)-3-(4-p-tolylpiperazin-1-yl)propan-1-amine NA 130010 NA NA NA NA BindingDB|TTD
CACNA1H N-[[4-(3-aminopropoxy)phenyl]methyl]-N-methyl-6-[3-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid NA 239000 NA NA NA NA TTD
CACNA1H N-[[4-(3-aminopropoxy)phenyl]methyl]-6-(4-fluorophenoxy)-N-methyl-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid NA 492000 NA NA NA NA TTD