| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CACNA1H |
2-[3-[4-[[Methyl-[6-[3-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-yl]amino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
771000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
2-[3-[4-[[[6-(4-Fluorophenoxy)-1,3-benzothiazol-2-yl]amino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
288000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
N-[[4-(3-aminopropoxy)phenyl]methyl]-6-[4-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid |
NA |
112000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
N-[[4-[3-(dimethylamino)propoxy]phenyl]methyl]-6-[3-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid |
NA |
110000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
2,2,2-Trifluoroacetic acid;2-[3-[4-[[[6-[3-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-yl]amino]methyl]phenoxy]propyl]guanidine |
NA |
270000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
2-[3-[4-[[(6-Phenoxy-1,3-benzothiazol-2-yl)amino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
166000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
4-[[2-[[4-(3-Aminopropoxy)phenyl]methylamino]-1,3-benzothiazol-6-yl]oxy]phenol;2,2,2-trifluoroacetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
4-[[2-[[4-(3-Aminopropoxy)phenyl]methyl-methylamino]-1,3-benzothiazol-6-yl]oxy]benzonitrile;2,2,2-trifluoroacetic acid |
NA |
328000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
2-[3-[4-[[[6-(4-Hydroxyphenoxy)-1,3-benzothiazol-2-yl]-methylamino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
332000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
2-[3-[4-[[[6-(4-Hydroxyphenoxy)-1,3-benzothiazol-2-yl]amino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
319000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
N-[[4-(3-aminopropoxy)phenyl]methyl]-N-methyl-6-[4-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid |
NA |
248000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
2,2,2-Trifluoroacetic acid;2-[3-[4-[[[6-[4-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-yl]amino]methyl]phenoxy]propyl]guanidine |
NA |
195000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
2-[3-[4-[[[6-(4-Cyanophenoxy)-1,3-benzothiazol-2-yl]-methylamino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
153000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
2-[3-[4-[[Methyl-[6-[4-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-yl]amino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
212000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
N-[[4-(3-aminopropoxy)phenyl]methyl]-6-(4-fluorophenoxy)-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid |
NA |
688000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
N-[[4-(3-aminopropoxy)phenyl]methyl]-6-[3-(trifluoromethyl)phenoxy]-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid |
NA |
171000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
N-[[4-[3-(dimethylamino)propoxy]phenyl]methyl]-6-(4-fluorophenoxy)-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
4-[[2-[[4-(3-Aminopropoxy)phenyl]methyl-methylamino]-1,3-benzothiazol-6-yl]oxy]phenol;2,2,2-trifluoroacetic acid |
NA |
165000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
2-[3-[4-[[[6-(4-Fluorophenoxy)-1,3-benzothiazol-2-yl]-methylamino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
521000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
2-[3-[4-[[Methyl-(6-phenoxy-1,3-benzothiazol-2-yl)amino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
498000 |
NA |
NA |
NA |
NA |
TTD |