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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CACNA1S Procainamide NA 389500 NA NA NA NA PubChem
CACNA1S Sotalol NA 193300 NA NA NA NA PubChem
CACNA1S Raltegravir NA 246700 NA NA NA NA PubChem
CACNA1S Ceftriaxone NA 153800 NA NA NA NA PubChem
CACNA1S Voriconazole NA 414200 NA NA NA NA PubChem
CALCRL deamino-hPhe-Tyr(3,5-diBr)-Lys-NHEtPh NA 300000 NA NA NA NA TTD
CALCRL deamino-hPhe-D-Tyr(3,5-diBr)-D-Lys-NHEtPh NA 300000 NA NA NA NA TTD
CALCRL N-{(S)-2-(4-Amino-3,5-dibromo-phenyl)-1-[(R)-5-amino-1-(4-phenyl-piperazine-1-carbonyl)-pentylcarbamoyl]-ethyl}-4-phenyl-butyramide NA 300000 NA NA NA NA TTD
CALCRL N-{(S)-2-(4-Amino-3,5-dibromo-phenyl)-1-[(R)-5-amino-1-(piperazine-1-carbonyl)-pentylcarbamoyl]-ethyl}-4-phenyl-butyramide NA 300000 NA NA NA NA TTD
CALCRL (2R)-6-amino-2-[[(2S)-3-(4-amino-3,5-dibromophenyl)-2-(3-phenylpropanoylamino)propanoyl]amino]-N-(2-phenylethyl)hexanamide NA 196000 NA NA NA NA TTD
CALM1 Flavone NA 102280 NA NA NA NA PubChem
CALM1 Clozapine NA 140000 NA NA NA NA PubChem
CALM2 Flavone NA 102280 NA NA NA NA PubChem
CALM2 Clozapine NA 140000 NA NA NA NA PubChem
CALM3 Flavone NA 102280 NA NA NA NA PubChem
CALM3 Clozapine NA 140000 NA NA NA NA PubChem
CAMK2A MLCK inhibitor peptide 18 NA 200000 NA NA NA NA TTD
CAMK2A R-K-K-Y-(Ach)-Y-R-R-K-NH2 NA 200000 NA NA NA NA TTD
CAMK2A R-K-K-Y-K-P-R-R-K-NH2 NA 200000 NA NA NA NA TTD
CAMK2A R-K-K-Y-K-N-R-R-K-NH2 NA 200000 NA NA NA NA TTD