| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CACNA1H |
4-[[2-[[4-(3-Aminopropoxy)phenyl]methylamino]-1,3-benzothiazol-6-yl]oxy]benzonitrile;2,2,2-trifluoroacetic acid |
NA |
109000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
N-[[4-(3-aminopropoxy)phenyl]methyl]-6-phenoxy-1,3-benzothiazol-2-amine;2,2,2-trifluoroacetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
2-[3-[4-[[[6-(4-Cyanophenoxy)-1,3-benzothiazol-2-yl]amino]methyl]phenoxy]propyl]guanidine;2,2,2-trifluoroacetic acid |
NA |
326000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
6-[({1-[2-(7-Methoxy-2-oxoquinoxalin-1(2H)-yl)ethyl]piperidin-4-yl}amino)methyl]-2H-pyrido[3,2-b][1,4]oxazin-3(4H)-one |
NA |
333000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1H |
Benzo[b][1]benzazepin-11-yl-[4-[3-(dimethylamino)propoxy]phenyl]methanone |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB |
| CACNA1H |
5,6-Dihydrobenzo[b][1]benzazepin-11-yl-[4-[3-(dimethylamino)propoxy]phenyl]methanone |
NA |
108000 |
NA |
NA |
NA |
NA |
BindingDB |
| CACNA1H |
6-((((1R,4r)-4-((R)-1-Amino-2-(7-methoxy-2-oxo-1,5-naphthyridin-1(2H)-yl)ethyl)cyclohexyl)amino)methyl)-2H-pyrido[3,2-b][1,4]oxazin-3(4H)-one |
NA |
333000 |
NA |
NA |
NA |
NA |
TTD |
| CACNA1I |
N-[(4-fluorophenyl)methyl]-2-[3-phenyl-2-(5-pyrrolidin-1-ylpentylsulfanyl)-4H-quinazolin-4-yl]acetamide |
NA |
663900 |
NA |
NA |
NA |
NA |
BindingDB |
| CACNA1I |
Ethosuximide |
NA |
5000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| CACNA1S |
Paliperidone |
NA |
193900 |
NA |
NA |
NA |
NA |
PubChem |
| CACNA1S |
Acetic acid 4-(4-methoxymethoxy-phenyl)-1-(2-methylamino-ethyl)-2-oxo-6-trifluoromethyl-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl ester |
NA |
NA |
155000 |
NA |
NA |
NA |
BindingDB |
| CACNA1S |
Moxifloxacin |
NA |
173000 |
NA |
NA |
NA |
NA |
PubChem |
| CACNA1S |
Telbivudine |
NA |
713900 |
NA |
NA |
NA |
NA |
PubChem |
| CACNA1S |
Disopyramide |
NA |
1036700 |
NA |
NA |
NA |
NA |
PubChem |
| CACNA1S |
Ribavirin |
NA |
622500 |
NA |
NA |
NA |
NA |
PubChem |
| CACNA1S |
Metronidazole |
NA |
177900 |
NA |
NA |
NA |
NA |
PubChem |
| CACNA1S |
Piperacillin |
NA |
1226000 |
NA |
NA |
NA |
NA |
PubChem |
| CACNA1S |
Sitagliptin |
NA |
147100 |
NA |
NA |
NA |
NA |
PubChem |
| CACNA1S |
Linezolid |
NA |
105400 |
NA |
NA |
NA |
NA |
PubChem |
| CACNA1S |
Pentobarbital |
NA |
299000 |
NA |
NA |
NA |
NA |
PubChem |