| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CASP6 |
(S)-1-(4-iodobenzyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
(S)-1-(4-methoxybenzyl)-5-[1-(2-methoxymethylpyrrolidinyl)-sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
(S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1-methylindoline-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
(S)-1-(4-(2-(4-methylphenylsulfonyloxy)ethoxy)benzyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
(S)-1-(4-(tert-butyldimethylsilyloxy)benzyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
(S)-1-(4-(2-bromoethoxy)benzyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
(S)-5-[1-(2-phenoxymethylpyrrolidinyl)sulfonyl]-1-(4-(tributylstannyl)benzyl)isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
2-[4-[[2,3-dioxo-5-[(2S)-2-(phenoxymethyl)pyrrolidin-1-yl]sulfonylindol-1-yl]methyl]phenoxy]ethyl 4-methylbenzenesulfonate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
(S)-1-(4-(tert-butyldimethylsilyloxy)benzyl)-5-[1-(2-phenoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
(S)-1-(4-(2-bromoethoxy)benzyl)-5-[1-(2-phenoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
(S)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]-1-(4-(tributylstannyl)benzyl)isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
1-butyl-7-iodo-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP6 |
1-(4-fluorobutyl)-7-iodo-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP6 |
1-(4-hydroxybutyl)-7-iodo-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP6 |
7-bromo-1-(4-hydroxybutyl)-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP6 |
7-chloro-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP6 |
1-butyl-7-chloro-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP6 |
7-chloro-1-(3-fluoropropyl)-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP6 |
7-fluoro-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP6 |
5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1-[2-(oxiran-2-yl)ethyl]indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |