| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CASP6 |
5-[2-(3-methoxypropyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
1-Butyl-5-[2-(3-methoxypropyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
1-(4-Fluorobutyl)-5-[2-(3-methoxypropyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
5-[(2S)-2-(ethoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
5-[(2S)-2-(ethoxymethyl)pyrrolidin-1-yl]sulfonyl-1-(4-fluorobutyl)indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
5-[(2S)-2-(2-fluoroethoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
1-butyl-5-[(2S)-2-(2-fluoroethoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
1-(4-fluorobutyl)-5-[(2S)-2-(2-fluoroethoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
5-[(2S)-2-(2,2,2-trifluoroethoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
1-butyl-5-[(2S)-2-(2,2,2-trifluoroethoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
1-(4-fluorobutyl)-5-[(2S)-2-(2,2,2-trifluoroethoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP6 |
Caspase-3/7 Inhibitor I |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB |
| CASP7 |
7-iodo-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP7 |
7-bromo-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP7 |
7-chloro-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP7 |
N-(2-hydroxy-1-methylindol-3-yl)imino-6-(4-methoxyphenyl)-2-methylpyridine-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
N-(2-hydroxy-1-methylindol-3-yl)imino-6-(3-methoxyphenyl)-2-methylpyridine-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
N-(2-hydroxy-1-methylindol-3-yl)imino-6-(2-methoxyphenyl)-2-methylpyridine-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
6-(3,4-dimethoxyphenyl)-N-(2-hydroxy-1-methylindol-3-yl)imino-2-methylpyridine-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
6-(4-fluorophenyl)-N-(2-hydroxy-1-methylindol-3-yl)imino-2-methylpyridine-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |