| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CASP7 |
N-(2-hydroxy-1-methylindol-3-yl)imino-2-methyl-6-(2-nitrophenyl)pyridine-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
6-(3-chlorophenyl)-N-(2-hydroxy-1-methylindol-3-yl)imino-2-methylpyridine-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
1,2-Benzisothiazoline-3-one |
NA |
137400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP7 |
2-(2,3-Dihydro-1,4-benzodioxin-2-yl)-1,3-thiazole-4-carboxylic acid |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP7 |
[2-(2,3-Dihydro-1,4-benzodioxin-2-yl)-1,3-thiazol-4-yl](thiophen-2-ylsulfanyl)methanone |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
4-{[2-(2,3-Dihydro-1,4-benzodioxin-2-yl)-1,3-thiazol-4-yl]carbonyl}morpholine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
2-(2,3-dihydro-1,4-benzodioxin-2-yl)-N,N-dimethyl-1,3-thiazole-4-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
2-(2,3-dihydro-1,4-benzodioxin-2-yl)-N-(furan-2-ylmethyl)-1,3-thiazole-4-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
(4-Chlorophenyl) 2-(2,3-dihydro-1,4-benzodioxin-3-yl)-1,3-thiazole-4-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
Phenyl 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-1,3-thiazole-4-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
Ethyl 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4-methyl-1,3-thiazole-5-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
2-(2,3-Dihydro-1,4-benzodioxin-2-yl)-4-methyl-1,3-thiazole-5-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
(S)-1-[3-(3-Hydroxypropoxy)propyl]-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
113000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP7 |
(S)-3-(((9H-fluoren-9-yl)methoxy)carbonylamino)-5-(phenylsulfonyl)pent-4-enoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
(S)-3-(((9H-fluoren-9-yl)methoxy)carbonylamino)-5-(methylsulfonyl)pent-4-enoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
(S)-3-((2S,3S)-2-(benzyloxycarbonylamino)-3-methylpentanamido)-5-(phenylsulfonyl)pent-4-enoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
(S)-3-((2S,3S)-2-(benzyloxycarbonylamino)-3-methylpentanamido)-5-(methylsulfonyl)pent-4-enoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
(S)-3-((S)-2-(((9H-fluoren-9-yl)methoxy)carbonylamino)-3-methylbutanamido)-5-(phenylsulfonyl)pent-4-enoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
(S)-3-((S)-2-(((9H-fluoren-9-yl)methoxy)carbonylamino)-3-methylbutanamido)-5-(methylsulfonyl)pent-4-enoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
(S)-3-((S)-2-(benzyloxycarbonylamino)-3-methylbutanamido)-5-(methylsulfonyl)pent-4-enoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |