| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CASP8 |
(S)-1-(4-(2-bromoethoxy)benzyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
(S)-5-[1-(2-phenoxymethylpyrrolidinyl)sulfonyl]-1-(4-(tributylstannyl)benzyl)isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
2-[4-[[2,3-dioxo-5-[(2S)-2-(phenoxymethyl)pyrrolidin-1-yl]sulfonylindol-1-yl]methyl]phenoxy]ethyl 4-methylbenzenesulfonate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
(S)-1-(4-(tert-butyldimethylsilyloxy)benzyl)-5-[1-(2-phenoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
(S)-1-(4-(2-bromoethoxy)benzyl)-5-[1-(2-phenoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
(S)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]-1-(4-(tributylstannyl)benzyl)isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
4-{[2-(2,3-Dihydro-1,4-benzodioxin-2-yl)-1,3-thiazol-4-yl]carbonyl}morpholine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
2-(2,3-dihydro-1,4-benzodioxin-2-yl)-N,N-dimethyl-1,3-thiazole-4-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
(4-Chlorophenyl) 2-(2,3-dihydro-1,4-benzodioxin-3-yl)-1,3-thiazole-4-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
Ethyl 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4-methyl-1,3-thiazole-5-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
2-(2,3-Dihydro-1,4-benzodioxin-2-yl)-4-methyl-1,3-thiazole-5-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
1-benzyl-3,7-dimethyl-8-sulfanylidene-9H-purine-2,6-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
H-Ala-Met-Val-Gly-Arg-Cys(1)-Tyr-D-Arg-Pro-Cys(1)-D-Trp-D-Glu-D-Val-OH |
NA |
NA |
NA |
25000000 |
NA |
NA |
TTD |
| CASP8 |
H-D-Cys(1)-Gly-Arg-D-Val-Tyr-D-Arg-Pro-Cys(1)-D-Trp-D-Glu-D-Val-OH |
NA |
NA |
NA |
4000000 |
NA |
NA |
TTD |
| CASP8 |
(S)-1-(4-hydroxybenzyl)-5-[1-(2-methoxymethylpyrrolidinyl)-sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
1-ethyl-8-mercapto-3,7-dimethyl-1H-purine-2,6(3H,7H)-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
H-Asp-Thr-Met-Arg-Ala-Met-D-Cys(1)-Gly-Arg-Val-Tyr-Arg-Pro-Cys(1)-Trp-Glu-Val-OH |
NA |
NA |
NA |
25000000 |
NA |
NA |
TTD |
| CASP8 |
Caffeine, 8-mercapto- |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CBS |
sodium;[(1S)-1-methyl-12,17-dioxo-14-oxapentacyclo[11.6.1.02,11.04,9.016,20]icosa-2(11),3,5,7,9,13(20),15-heptaen-5-yl] sulfate |
NA |
136000 |
NA |
NA |
NA |
NA |
TTD |
| CBS |
5-Benzylidene-2-thiohydantoin |
NA |
170000 |
NA |
NA |
NA |
NA |
TTD |