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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CBX7 Ac-Phe-Ala-Leu-Lys(Me3)-DL-Nva-ol NA 500000 NA NA NA NA TTD
CBX7 [(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-[[(1S,2S)-2-hydroxycyclohexyl]amino]-6-oxohexyl]-trimethylazanium NA 250000 NA NA NA NA TTD
CBX7 Ac-Phe-Ala-Leu-Lys(Me3)-Ac5c-ol NA 250000 NA NA NA NA TTD
CBX7 Ac-Phe-Ala-Leu-Lys(Me3)-NHPr NA 102000 NA NA NA NA TTD
CBX7 [(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-[2-[(2-methylpropan-2-yl)oxycarbonylamino]ethylamino]-6-oxohexyl]-trimethylazanium NA 105000 NA NA NA NA TTD
CBX7 Bes(4-OMe)-Ala-Leu-Lys(Me3)-Ser-NH2 NA 250000 NA NA NA NA TTD
CBX7 [(5S)-6-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-4-methyl-2-[[(2S)-2-(pyridin-3-ylsulfonylamino)propanoyl]amino]pentanoyl]amino]-6-oxohexyl]-trimethylazanium NA 250000 NA NA NA NA TTD
CBX7 [(5S)-6-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-2-[[(2S)-2-[(4-carboxyphenyl)methylamino]propanoyl]amino]-4-methylpentanoyl]amino]-6-oxohexyl]-trimethylazanium NA 2000000 NA NA NA NA TTD
CBX7 Bn-Ala-Leu-Lys(Me3)-Ser-NH2 NA 2000000 NA NA NA NA TTD
CBX7 Tos-Phe-Ala-Leu-Lys(Me3)-Ser-NH2 NA 250000 NA NA NA NA TTD
CCKAR Imipenem NA NA NA NA NA 300000 PubChem
CCKAR H-Asp-Tyr(SO3H)-Met-Dap(1)-Trp-Met-Asp-Phe-Ala-(1) NA 1000000 NA NA NA NA TTD
CCKAR Cefazolin NA NA NA NA NA 300000 PubChem
CCKAR Meropenem NA NA NA NA NA 300000 PubChem
CCKAR Cefepime NA NA NA NA NA 300000 PubChem
CCKAR Ceftazidime NA NA NA NA NA 300000 PubChem
CCKAR Aztreonam NA NA NA NA NA 400000 PubChem
CCKAR Carumonam NA NA NA NA NA 500000 PubChem
CCKAR Doripenem NA NA NA NA NA 300000 PubChem
CCKBR beta-Carboline-3-carboxylic acid methyl ester NA 150000 NA NA NA NA BindingDB|TTD