| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CCKBR |
CCK-A Agonist 18 |
NA |
173780.08 |
NA |
NA |
NA |
NA |
TTD |
| CCKBR |
N-(2-oxo-5-phenyl-1,3-dihydro-1,4-benzodiazepin-3-yl)-2,3-dihydro-1H-indole-2-carboxamide |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CCKBR |
2-chloro-N-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]benzamide |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CCKBR |
3,5-Dichloro-N-(2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-benzamide |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CCKBR |
4-methyl-N-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]pentanamide |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CCKBR |
N-(9H-beta-Carbolin-3-yl)-benzamide |
NA |
223000 |
NA |
NA |
NA |
NA |
BindingDB |
| CCKBR |
(1-[(3-[(2,3-dihydro-2-oxo-5-phenyl-1,4-benzodiazepin-3-yl)methyl]-2,3-dihydro-1H-indol-1-yl) carbonyl]-3-methylbutyl]-carbamic acid-1,1-dimethylethyl ester |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CCKBR |
N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-4-(4-methyl-piperazin-1-yl)-4-oxo-butyl]-3,5-dichloro-benzamide; hydrochloride |
NA |
120500 |
NA |
NA |
NA |
NA |
BindingDB |
| CCKBR |
N-{1-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-pentyl}-3-(3-phenyl-propionylamino)-succinamic acid |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CCKBR |
3-Chloro-N-[1-(3,3-dimethyl-butylcarbamoyl)-4-(4-methyl-piperazin-1-yl)-4-oxo-butyl]-benzamide; hydrochloride |
NA |
103800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CCKBR |
Proglumide |
NA |
900000|2500000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| CCKBR |
1-methyl-3-[[(3S)-1-methyl-2,3-dihydroindol-3-yl]methyl]-5-phenyl-3H-1,4-benzodiazepin-2-one |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CCKBR |
(4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-6-(pent-4-ynoylamino)hexanoyl]amino]-3-hydroxypropanoyl]amino]hexanoyl]amino]-5-[[(2S)-1-[[(2R)-1-[[(2S)-1-[[(2S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-5-oxopentanoic acid |
NA |
4600000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CCL2 |
nonasodium;(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-5-acetamido-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-5-acetamido-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6S)-5-acetamido-4-hydroxy-6-pentoxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-3,4-dihydroxy-5-sulfonatooxyoxane-2-carboxylate |
NA |
NA |
250000000 |
NA |
NA |
NA |
BindingDB |
| CCL2 |
nonasodium;(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6S)-6-(5-aminopentoxy)-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-3,4-dihydroxy-5-sulfonatooxyoxane-2-carboxylate |
NA |
NA |
250000000 |
NA |
NA |
NA |
BindingDB |
| CCL5 |
nonasodium;(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-5-acetamido-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4R,5R,6S)-5-acetamido-4-hydroxy-6-pentoxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-2-carboxylato-4,5-dihydroxyoxan-3-yl]oxy-4-hydroxy-5-(sulfonatoamino)-2-(sulfonatooxymethyl)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-3,4-dihydroxy-5-sulfonatooxyoxane-2-carboxylate |
NA |
NA |
25000000 |
NA |
NA |
NA |
BindingDB |
| CCL5 |
nonasodium;(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-5-acetamido-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-5-acetamido-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6S)-5-acetamido-4-hydroxy-6-pentoxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(sulfonatooxymethyl)oxan-3-yl]oxy-3,4-dihydroxy-5-sulfonatooxyoxane-2-carboxylate |
NA |
NA |
25000000 |
NA |
NA |
NA |
BindingDB |
| CCL5 |
nonasodium;(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6S)-6-(5-aminopentoxy)-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-3,4-dihydroxy-5-sulfonatooxyoxane-2-carboxylate |
NA |
NA |
25000000 |
NA |
NA |
NA |
BindingDB |
| CCNB1 |
Genistein |
NA |
370000 |
NA |
NA |
NA |
NA |
PubChem |
| CCND1 |
N-(6-methoxyquinolin-8-yl)-N',N'-bis(3-methylbutyl)propane-1,3-diamine |
NA |
325000 |
NA |
NA |
NA |
NA |
BindingDB |