| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CCR1 |
4,7-Dimethyl-1,10-phenanthroline |
NA |
112000 |
NA |
NA |
NA |
NA |
BindingDB |
| CCR1 |
3,4,7,8-Tetramethyl-1,10-phenanthroline |
NA |
158489.32|171000 |
NA |
NA |
NA |
NA |
BindingDB |
| CCR1 |
4-Methyl-1,10-phenanthroline |
NA |
251188.64|261000 |
NA |
NA |
NA |
NA |
BindingDB |
| CCR3 |
N-{1-[4-(3,4-Dichloro-benzyl)-cyclohexylmethyl]-2-methyl-propyl}-4-methyl-benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CCR3 |
N-[1-(1-Benzyl-piperidin-4-ylmethyl)-2-methyl-propyl]-4-methyl-benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CCR4 |
2-amino-N-((2S,3R)-1-(2,6-dioxopiperidin-3-ylamino)-3-methyl-1-oxopentan-2-yl)benzamide |
NA |
836000 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
4-[4-[[(3R)-1-butyl-3-[(1R)-1-hydroxy-2-methylpropyl]-2,5-dioxo-1,4,9-triazaspiro[5.5]undecan-9-yl]methyl]phenoxy]benzoic acid |
NA |
229000 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
10-Methoxydihydrofuscin |
NA |
154000 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
N-[[5,7-dimethyl-8-[[[4-(trifluoromethyl)benzoyl]amino]methyl]-2,3-dihydro-1H-indolizin-4-ium-6-yl]methyl]-4-(trifluoromethyl)benzamide;chloride |
NA |
121500 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
4-cyano-N-[[8-[[(4-cyanobenzoyl)amino]methyl]-5,7-dimethyl-2,3-dihydro-1H-indolizin-4-ium-6-yl]methyl]benzamide;chloride |
NA |
101200 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
4-amino-N-[[8-[[(4-aminobenzoyl)amino]methyl]-5,7-dimethyl-2,3-dihydro-1H-indolizin-4-ium-6-yl]methyl]benzamide;chloride |
NA |
173900 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
N-[4-[5-(3,4-dihydroxyphenyl)-3-oxo-pentyl]phenyl]-4-methoxy-benzamide |
NA |
NA |
NA |
200000 |
NA |
NA |
TTD |
| CCR5 |
Abametapir |
NA |
199526|206000 |
NA |
NA |
NA |
NA |
PubChem |
| CCR5 |
6,6'-Bi-2-picoline |
NA |
501187.23 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
1,10-Phenanthroline-2,9-diyldimethanol |
NA |
587000 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
2,9-Bis(bromomethyl)-1,10-phenanthroline |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
4-[4-[[(3R)-3-[(R)-cyclohexyl(hydroxy)methyl]-1-(3-hydroxybutyl)-2,5-dioxo-1,4,9-triazaspiro[5.5]undecan-9-yl]methyl]phenoxy]-N-methylbenzamide |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
4-[4-[[(3R)-3-[(R)-cyclohexyl(hydroxy)methyl]-2,5-dioxo-1-(2,2,2-trifluoroethyl)-1,4,9-triazaspiro[5.5]undecan-9-yl]methyl]phenoxy]-N-methylbenzamide |
NA |
1148000 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
4-[4-[[(3R)-3-[(R)-cyclohexyl(hydroxy)methyl]-1-heptyl-2,5-dioxo-1,4,9-triazaspiro[5.5]undecan-9-yl]methyl]phenoxy]-N-methylbenzamide |
NA |
190000 |
NA |
NA |
NA |
NA |
TTD |
| CCR5 |
4-[4-[[(3R)-3-[(R)-cyclohexyl(hydroxy)methyl]-2,5-dioxo-1-(2,2,3,3,3-pentafluoropropyl)-1,4,9-triazaspiro[5.5]undecan-9-yl]methyl]phenoxy]-N-methylbenzamide |
NA |
270000 |
NA |
NA |
NA |
NA |
TTD |