| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CCND1 |
(2S)-2-[bis(2-methylpropyl)amino]-1-[(6-methoxy-2-methylquinolin-8-yl)amino]propan-2-ol |
NA |
691000 |
NA |
NA |
NA |
NA |
BindingDB |
| CCND1 |
5-chloro-N-(3,4-dichlorophenyl)-2-methylbenzenesulfonamide |
NA |
110400 |
NA |
NA |
NA |
NA |
BindingDB |
| CCND1 |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
NA |
129000 |
NA |
NA |
NA |
NA |
BindingDB |
| CCND1 |
4-Phenyl-[1]benzofuro[2,3-b]pyridine-3,6-diol |
773000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CCND1 |
Genistein |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| CCND1 |
Triamterene |
NA |
210000 |
NA |
NA |
NA |
NA |
PubChem |
| CCND1 |
4-methyl-N-[3-(trifluoromethyl)phenyl]benzenesulfonamide |
NA |
208800 |
NA |
NA |
NA |
NA |
BindingDB |
| CCNE1 |
Alvocidib |
NA |
330000 |
NA |
NA |
NA |
NA |
PubChem |
| CCNE2 |
Alvocidib |
NA |
330000 |
NA |
NA |
NA |
NA |
PubChem |
| CCNT1 |
N-(2-(1H-indol-3-yl)ethyl)-4-chloro-N-methylbenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CCNT1 |
N-[2-(1H-Indol-3-yl)ethyl]-N-methyl-4-phenylbenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CCNT1 |
N-(2-(1H-indol-3-yl)ethyl)-4-tert-butyl-N-methylbenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CCNT1 |
2-ethyl-N-[5-(4-hydroxyphenyl)-2H-pyrazolo[3,4-b]pyridin-3-yl]butanamide |
NA |
529300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CCNT1 |
Fascaplysine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| CCR1 |
4,4'-Dimethyl-2,2'-bipyridine |
NA |
101000 |
NA |
NA |
NA |
NA |
BindingDB |
| CCR1 |
2,2'-Bipyridine |
NA |
125892.54|126000 |
NA |
NA |
NA |
NA |
BindingDB |
| CCR1 |
Abametapir |
NA |
199526.23|204000|199526 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| CCR1 |
4,4'-Dimethoxy-2,2'-bipyridyl |
NA |
179000|199526.23 |
NA |
NA |
NA |
NA |
BindingDB |
| CCR1 |
1,10-Phenanthroline-2,9-diyldimethanol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CCR1 |
5-Methyl-1,10-phenanthroline |
NA |
119000|125892.54 |
NA |
NA |
NA |
NA |
BindingDB |