| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CASP7 |
5-[(2S,5R)-2,5-bis(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
5-[(2S,5S)-2,5-bis(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
5-[(2S,4R)-4-methoxy-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
5-[(2S,4S)-4-methoxy-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
1-butyl-5-[(2S,4S)-4-methoxy-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
5-[(2S,4R)-2-(methoxymethyl)-4-(trifluoromethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
1-(4-fluorobutyl)-5-[(2S,4S)-2-(methoxymethyl)-4-(trifluoromethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
147000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP7 |
5-[(2R,5S)-2,5-bis(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1-butylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
5-[(2R,5S)-2,5-bis(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1-(4-fluorobutyl)indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
5-[(2S,4S)-4-[2-[2-[2-(2-hydroxyethoxy)ethoxy]ethoxy]ethoxy]-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
1-butyl-5-[(2S,4S)-4-[2-[2-[2-(2-hydroxyethoxy)ethoxy]ethoxy]ethoxy]-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
5-[(2S,4R)-4-[2-[2-[2-(2-hydroxyethoxy)ethoxy]ethoxy]ethoxy]-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP7 |
N-[(4-morpholin-4-ylphenyl)methyl]-3-oxo-1,2-benzothiazole-2-carboxamide |
NA |
248000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP7 |
Miristalkonium chloride |
NA |
NA |
NA |
NA |
25118900 |
NA |
PubChem |
| CASP7 |
N-(4-morpholin-4-ylphenyl)-2-(3-oxo-1,2-benzothiazol-2-yl)acetamide |
NA |
100400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP8 |
(S)-1-(4-iodobenzyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
(S)-1-(4-methoxybenzyl)-5-[1-(2-methoxymethylpyrrolidinyl)-sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
(S)-5-(2-(methoxymethyl)pyrrolidin-1-ylsulfonyl)-1-methylindoline-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
(S)-1-(4-(2-(4-methylphenylsulfonyloxy)ethoxy)benzyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP8 |
(S)-1-(4-(tert-butyldimethylsilyloxy)benzyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |