| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CDK2 |
5-Hydroxynaphthalene-1-sulfonamide |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
4-[(2,6-dichlorobenzoyl)amino]-N-[1-(2,6-dichlorobenzoyl)piperidin-4-yl]-1H-pyrazole-5-carboxamide |
NA |
760200 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK2 |
1H-Indazole |
NA |
185000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
[4-Amino-2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-5-thiazolyl](2,3-dihydro-1,4-benzodioxin-6-yl)methanone |
NA |
2360000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK2 |
[4-Amino-2-[[4-[4-(1-methylethyl)-1-piperazinyl]phenyl]amino]-5-thiazolyl](3-methoxyphenyl)methanone |
NA |
4144000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK2 |
7-(Dimethylamino)-3,6,6-trimethyl-1-pyridin-2-yl-5,7-dihydroindazol-4-one |
NA |
630000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK2 |
7-Phenylsulfonyl-1-(2-pyridyl)-3,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydroindazole |
NA |
107000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK2 |
5-(4-Hydroxy-phenylamino)-2-methyl-benzothiazole-4,7-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CDK4 |
1-[2-(1H-Indol-3-yl)-ethyl]-5-methyl-1H-indole |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
3-(2-Indol-1-yl-ethyl)-5-methyl-1H-indole |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
5-Chloro-1-[2-(1H-indol-3-yl)-ethyl]-1H-indole |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
N-(2-(1H-indol-3-yl)ethyl)-N,2-dimethylbenzamide |
NA |
113000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
N-(2-(1H-indol-3-yl)ethyl)-2-fluoro-N-methylbenzamide |
NA |
103000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
N-(2-(1H-indol-3-yl)ethyl)-3-chloro-N-methylbenzamide |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3R,4R)-4-hydroxy-1-methylpiperidin-3-yl]chromen-4-one |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3R,4S)-4-hydroxy-1-methylpiperidin-3-yl]chromen-4-one |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
2-(2-Chloro-phenyl)-5,7-dihydroxy-8-pyrimidin-5-yl-chromen-4-one |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
1-(2,3-Dihydro-indol-1-yl)-2-(5-fluoro-1H-indol-3-yl)-ethane-1,2-dione |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
1-(5-Fluoro-2,3-dihydro-indol-1-yl)-2-(1H-indol-3-yl)-ethane-1,2-dione |
NA |
136000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
N-[5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl]-5-fluoro-4-(4-fluoro-7,8,9,10-tetrahydro-6H-azepino[1,2-a]benzimidazol-2-yl)pyrimidin-2-amine |
NA |
147300 |
NA |
NA |
NA |
NA |
BindingDB |