Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CDK4 | US10696678, Example 17 | NA | 235600 | NA | NA | NA | NA | BindingDB |
| CDK4 | 7H-Pyrido(4,3-c)carbazole | NA | 159000 | NA | NA | NA | NA | BindingDB |
| CDK4 | 7H-Pyrido(2,3-c)carbazole | NA | 197000 | NA | NA | NA | NA | BindingDB |
| CDK4 | 7H-Pyrido(3,2-c)carbazole | NA | 442000 | NA | NA | NA | NA | BindingDB |
| CDK4 | 6-(4-Methoxyphenyl)-4-[4-(4-methylpiperazin-1-yl)phenyl]-1,3-diphenylpyrazolo[3,4-b]pyridine-5-carbonitrile | NA | 104020 | NA | NA | NA | NA | BindingDB |
| CDK4 | 5-(1,3-Benzodioxol-5-ylmethylene)pyrimidine-2,4,6(1h,3h,5h)-trione | NA | 350000 | NA | NA | NA | NA | BindingDB |
| CDK4 | 6-(6-chloro-2H-chromen-3-yl)-1,3,5-triazine-2,4-diamine | NA | 450000 | NA | NA | NA | NA | BindingDB |
| CDK4 | 1-(1H-indol-3-yl)-2-(indolin-1-yl)ethane-1,2-dione | NA | 122000 | NA | NA | NA | NA | BindingDB |
| CDK4 | 9-Isopropyl-N*6*-(3-methyl-but-2-enyl)-9H-purine-2,6-diamine | NA | 200000 | NA | NA | NA | NA | BindingDB |
| CDK4 | 1,6-Bis-(indol-1-yl)-hexane | NA | 106000 | NA | NA | NA | NA | BindingDB |
| CDK4 | Olomoucine | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| CDK4 | N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine | NA | 376000 | NA | NA | NA | NA | BindingDB |
| CDK4 | Genistein | NA | 250000 | NA | NA | NA | NA | BindingDB|PubChem |
| CDK4 | Indenopyrazole 3f | NA | 108000 | NA | NA | NA | NA | BindingDB |
| CDK4 | NA | 240000 | NA | NA | NA | NA | BindingDB | |
| CDK4 | Diarylurea deriv. 1a | NA | 120000 | NA | NA | NA | NA | BindingDB |
| CDK4 | Diarylurea deriv. 1b | NA | 340000 | NA | NA | NA | NA | BindingDB |
| CDK4 | Diarylurea deriv. 1c | NA | 110000 | NA | NA | NA | NA | BindingDB |
| CDK4 | 1-Benzyl-3-(7-hydroxynaphthalen-1-yl)urea | NA | 410000 | NA | NA | NA | NA | BindingDB |
| CDK4 | 1-(7-Hydroxynaphthalen-1-yl)-3-propan-2-ylurea | NA | 220000 | NA | NA | NA | NA | BindingDB |