| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CDK4 |
Diarylurea deriv. 1g |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
Carbazole deriv. 18 |
NA |
605000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
N-tert-butyl-2-phenylquinazolin-4-amine |
NA |
361000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
Ethyl 4-(tert-butylamino)quinazoline-2-carboxylate |
NA |
168000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
4-Substituted quinazoline 24 |
NA |
119000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
Triamterene |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| CDK4 |
Methyl 4-hydroxy-2-{[4-hydroxy-3-(3-methylbut-2-en-1-yl)phenyl]methyl}-3-(4-hydroxyphenyl)-5-oxo-2,5-dihydrofuran-2-carboxylate |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
N-[(2S)-1-[[(2S)-1-[[4-(3-chlorophenoxy)pyridin-2-yl]methylamino]-4-methyl-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-1-(3,5-dichlorophenyl)-5-methyl-1,2,4-triazole-3-carboxamide |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
N-[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1-[[3-(3,5-dichlorophenoxy)phenyl]methylamino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]-1-(3,5-dichlorophenyl)-5-methyl-1,2,4-triazole-3-carboxamide |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[5-(imidazol-1-ylmethyl)furan-2-carbonyl]amino]pentanoyl]amino]-4-methylpentanoyl]amino]-3-methylpentanoyl]amino]-3-phenylpropanoic acid |
NA |
158600 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK4 |
(S)-methyl 4-hydroxy-2-(4-hydroxy-3-(3-methylbut-2-enyl)benzyl)-3-(4-hydroxyphenyl)-5-oxo-2,5-dihydrofuran-2-carboxylate |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK5 |
3-(6-Chloro-5-fluoro-1-methyl-1H-indol-3-yl)-4-(7-methoxybenzofuran-3-yl)pyrrole-2,5-dione |
NA |
108000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK5 |
|
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK5 |
Xanthen-9-one, 1.3 |
NA |
247000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK5 |
1,3,8-Trihydroxyxanthone |
NA |
533000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK5R1 |
6-Hydroxy-3-methoxy-4-phenylbenzo[4,3-b]pyridine |
217000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CDK5R1 |
1-[(4-methoxyphenyl)methyl]-3-[6-(2H-tetrazol-5-yl)-1,3-benzothiazol-2-yl]urea |
NA |
26400000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK6 |
N-[5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl]-5-fluoro-4-(5-fluoro-2,3-dihydro-1H-pyrrolo[1,2-a]benzimidazol-7-yl)pyrimidin-2-amine |
NA |
244100 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK6 |
5-fluoro-4-(5-fluoro-1,1-dimethyl-2,3-dihydropyrrolo[1,2-a]benzimidazol-7-yl)-N-[6-methyl-5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl]pyrimidin-2-amine |
NA |
271000 |
NA |
NA |
NA |
NA |
BindingDB |
| CDK6 |
4-(2-ethyl-5-fluoro-2,3-dihydro-1H-pyrrolo[1,2-a]benzimidazol-7-yl)-N-[5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl]-5-fluoropyrimidin-2-amine |
NA |
339000 |
NA |
NA |
NA |
NA |
BindingDB |