| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CETP |
N-[2-[[2-[2,2-dimethylpropanoyl(methyl)amino]phenyl]disulfanyl]phenyl]-N,2,2-trimethylpropanamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| CETP |
1,1,1-Trifluoro-3-((3-(3-methoxyphenoxy)phenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-ol |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(4-chloro-3-methylphenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-ol |
NA |
200032 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(4-isopropyl-3-methylphenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-ol |
NA |
200032 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
3-((3-(Biphenyl-4-yloxy)phenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)-1,1,1-trifluoropropan-2-ol |
NA |
2500345 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
1,1,1-Trifluoro-3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(4-(trifluoromethoxy)phenoxy)phenyl)amino)propan-2-ol |
NA |
400037 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
1,1,1-Trifluoro-3-((3-(4-propoxyphenoxy)phenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-ol |
NA |
400037 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(4-aminophenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-ol |
NA |
700003 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(2-chlorophenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-ol |
NA |
299985 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
1,1,1-Trifluoro-3-((3-(4-propylphenoxy)phenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-ol |
NA |
200032 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
1,1,1-Trifluoro-3-((3-(4-nitrophenoxy)phenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-ol |
NA |
500035 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(4-benzylphenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-ol |
NA |
2399938 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
(R)-3-((3-(4-chloro-3-ethylphenoxy)phenyl)(3-(trifluoromethoxy)benzyl)amino)-1,1,1-trifluoropropan-2-ol |
NA |
790000 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
(R)-3-((3-(4-chloro-3-ethylphenoxy)phenyl)(2-fluoro-4-(trifluoromethyl)benzyl)amino)-1,1,1-trifluoropropan-2-ol |
NA |
590000 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
1,1,1-Trifluoro-3-((3-(3-fluorophenoxy)phenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-ol |
NA |
299985 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
[2-[(1-Methylcyclohexanecarbonyl)amino]phenyl] 2-phenylacetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| CETP |
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(4-chlorophenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-ol |
NA |
299985 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
3-((3-(1,1,2,2-Tetrafluoroethoxy)benzyl)(3-(3,5-difluorophenoxy)phenyl)amino)-1,1,1-trifluoropropan-2-ol |
NA |
200032 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
Spongiadiol |
NA |
196000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CETP |
2,2-Dimethyl-thiopropionic acid 2-fluoro-6-[(1-methyl-cyclohexanecarbonyl)-amino]-phenyl ester |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |