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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CFD 5-fluoro-3-[(2-phenylcyclopropanecarbonyl)amino]-1H-indole-2-carboxylic acid NA|500000 NA 5e+05|NA NA NA NA ChEMBL|TTD
CFD 2-(3-Benzylureido)benzoic Acid NA|500000 NA 5e+05|NA NA NA NA ChEMBL|TTD
CFTR Tadalafil NA NA 175000 NA NA NA PubChem
CFTR 2-(1-Hydroxypentyl)-6-methyl-3-(2-phenylethyl)-1H-Indole-5-carboxylic acid NA 160000 NA NA NA NA TTD
CFTR 2-(4-carboxybutyl)-3-(hydroxymethyl)-5-methyl-1-phenethyl-1H-indole-6-carboxylic acid NA 170000 NA NA NA NA TTD
CFTR 7-Chlorobenzo[c]quinolizin-11-ium-6-ol;chloride NA NA NA 146000 NA NA TTD
CFTR 7-Chlorobenzo[c]quinolizin-11-ium-6-ol NA NA NA 146000 NA NA BindingDB
CFTR 2-(4-carboxy-1-hydroxybutyl)-6-methyl-3-phenethyl-1H-indole-5-carboxylic acid NA 330000 NA NA NA NA TTD
CFTR 2-((2-carboxyethyl)carbamoyl)-6-methyl-3-phenethyl-1H-indole-5-carboxylic acid NA 490000 NA NA NA NA TTD
CFTR Rescinnamine NA NA NA NA NA 142487 PubChem
CFTR Telmisartan NA NA 189300 NA NA NA PubChem
CFTR 10-Chloro-6-hydroxy-11lambda5-pyrido(1,2-A)quinolin-11-ylium chloride NA NA NA 141000 NA NA TTD
CFTR MPB-07 free acid NA NA NA 141000 NA NA BindingDB
CFTR 3-(hydroxymethyl)-5-methyl-2-pentyl-1-phenethyl-1H-indole-6-carboxylic acid NA 380000 NA NA NA NA TTD
CHAT 1-Anilino-8-naphthalenesulfonate 200000 NA NA NA NA NA BindingDB
CHAT 2-Anilinonaphthalene-6-sulfonic acid 800000 NA NA NA NA NA BindingDB
CHAT Naphthalene-1-sulfonate 1600000 NA NA NA NA NA BindingDB
CHAT 5-Phenylamino-naphthalene-1-sulfonic acid anion 1500000 NA NA NA NA NA BindingDB
CHAT 7-Phenylamino-naphthalene-1-sulfonic acid anion 150000 NA NA NA NA NA BindingDB
CHAT Adenosine Phosphate NA 1800000000000 NA NA NA NA PubChem