| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CETP |
2,2-Dimethyl-thiopropionic acid S-{3,5-difluoro-2-[(1-methyl-cyclohexanecarbonyl)-amino]-phenyl} ester |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| CETP |
2,2-Dimethyl-thiopropionic acid S-(4-methoxy-2-{[1-(3-methyl-butyl)-cyclohexanecarbonyl]-amino}-phenyl) ester |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| CETP |
2,2-Dimethyl-thiopropionic acid S-{4-methoxy-2-[(1-methyl-cyclohexanecarbonyl)-amino]-phenyl} ester |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| CETP |
2,2-Dimethyl-thiopropionic acid S-(4-methyl-2-{[1-(3-methyl-butyl)-cyclohexanecarbonyl]-amino}-phenyl) ester |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| CETP |
1,1,1-trifluoro-3-(5-(3-isopropylphenyl)-2-(3-(1,1,2,2-tetrafluoroethoxy)phenyl)-3,4-dihydroquinolin-1(2H)-yl)propan-2-ol |
NA |
277000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CETP |
1,1,1-trifluoro-3-(5-(3-isopropoxyphenyl)-2-(3-(1,1,2,2-tetrafluoroethoxy)phenyl)-3,4-dihydroquinolin-1(2H)-yl)propan-2-ol |
NA |
345000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CETP |
1,1,1-trifluoro-3-(2-(3-(1,1,2,2-tetrafluoroethoxy)phenyl)-5-(thiophen-2-yl)-3,4-dihydroquinolin-1(2H)-yl)propan-2-ol |
NA |
317000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CETP |
N,N'-(disulfanediyldibenzene-4,1-diyl)bis(2,2-dimethylpropanamide) |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CETP |
2,2-Dimethyl-thiopropionic acid S-{4-cyano-2-[(1-methyl-cyclohexanecarbonyl)-amino]-phenyl} ester |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CETP |
N-tert-butyl-2-[[2-(tert-butylcarbamoyl)phenyl]disulfanyl]benzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CETP |
2,2'-Dibenzoylaminodiphenyl disulfide |
NA |
101000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CETP |
(R)-1,1,1-trifluoro-3-((3-phenoxyphenyl)(3-(1,1,2,2-tetrafluoroethoxy)benzyl)amino)propan-2-ol |
NA |
640000 |
NA |
NA |
NA |
NA |
BindingDB |
| CETP |
Sphingosylphosphorylcholine |
NA |
156900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CETP |
Sulfiricin |
NA |
190000 |
NA |
NA |
NA |
NA |
TTD |
| CFD |
3-(((2-Carbamoyl-1H-indol-5-yl)oxy)methyl)benzoic acid |
NA |
NA |
1600000 |
NA |
NA |
NA |
ChEMBL |
| CFD |
N-[3'-(Aminomethyl)[1,1'-biphenyl]-3-yl]-3-methylbutanamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| CFD |
3-[3-(aminomethyl)phenyl]-N-benzylbenzamide |
NA |
310000 |
NA |
NA |
NA |
NA |
TTD |
| CFD |
N-[3-[3-(aminomethyl)phenyl]phenyl]benzamide |
NA |
257000 |
NA |
NA |
NA |
NA |
TTD |
| CFD |
N-[3-[3-(aminomethyl)phenyl]phenyl]acetamide |
NA |
690000 |
NA |
NA |
NA |
NA |
TTD |
| CFD |
N-[3-[3-(aminomethyl)phenyl]phenyl]-3-phenylpropanamide |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |