Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CTSD | US10246429, Example 247 | NA | 1192900 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 244 | NA | 150000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 288 | NA | 175000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 276 | NA | 156000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 267 | NA | 209000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 278 | NA | 199000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 175 | NA | 204000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 311 | NA | 681400|714000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 110 | NA | 403200 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 281 | NA | 269100 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 290 | NA | 400000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 233 | NA | 204000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 216 | NA | 390990 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 287 | NA | 205800 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 291 | NA | 290100 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 251 | NA | 360400 | NA | NA | NA | NA | BindingDB |
| CTSD | N-[(4S)-2-amino-3'-(3,6-dihydro-2H-pyran-5-yl)spiro[5H-1,3-oxazole-4,5'-chromeno[2,3-c]pyridine]-7'-yl]-5-chloropyridine-2-carboxamide | NA | 480000 | NA | NA | NA | NA | TTD |
| CTSD | US9611261, Example 28 | NA | 907850 | NA | NA | NA | NA | BindingDB |
| CTSD | US9611261, Example 141 | NA | 654540 | NA | NA | NA | NA | BindingDB |
| CTSD | US9611261, Example 142 | NA | 229080 | NA | NA | NA | NA | BindingDB |